SCHEMBL7112341

SCHEMBL7112341

CCCNc1cc[c]cc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
AR P10275 4/20 0.38
TLR7 Q9NYK1 1/20 0.36
PTPN1 P18031 1/20 0.34
IDO1 P14902 1/20 0.33
ALDH1A1 P00352 2/20 0.31
LIMK1 P53667 1/20 0.31
TRPA1 O75762 3/20 0.31
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7110018 0.86 PDE3B (0.36) PDE3BPDE3AAR
SCHEMBL7113956 0.79 TLR7 (0.40) PDE3BPDE3AARTLR7IDO1
SCHEMBL7447385 0.77 IDO1 (0.35) IDO1TRPA1
SCHEMBL6236003 0.75 POLB (0.50) PDE3BPDE3AARTLR7PTPN1
SCHEMBL7111154 0.74 TP53 (0.39) ALDH1A1CYP1A2POLB
SCHEMBL7113832 0.74 PDE3B (0.35) PDE3BPDE3AIDO1
SCHEMBL2209235 0.73 SLC22A12 (0.43) CYP1A2
SCHEMBL5217967 0.73 KMT2A (0.42) ALDH1A1CYP1A2POLB
SCHEMBL7112683 0.72 PDE3B (0.36) PDE3BPDE3AARTLR7
SCHEMBL687401 0.72 POLB (0.45) ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1351924-A2 DIAMINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Pharma Company (US) 2003-10-15 EP disclosed
WO-2002050019-A2 DIAMINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB PHARMA CO. (US) 2002-06-27 WO disclosed