SCHEMBL7113012

SCHEMBL7113012

Nc1c([N+](=O)[O-])cc(Cl)c(Cl)c1F.Nc1cc(Cl)c(Cl)c(F)c1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.46
CYP3A4 P08684 3/20 0.46
TSHR P16473 4/20 0.43
MAPT P10636 6/20 0.42
LMNA P02545 2/20 0.42
HPGD P15428 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
XBP1 P17861 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TLR9 Q9NR96 1/20 0.42
TDP1 Q9NUW8 4/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
PDE7A Q13946 1/20 0.39
ALOX15 P16050 1/20 0.38
HIF1A Q16665 1/20 0.38
TXNRD1 Q16881 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734435 0.93 TSHR (0.48) ALDH1A1CYP3A4TSHRMAPTLMNA
SCHEMBL7124662 0.92 ALDH1A1 (0.46) ALDH1A1CYP3A4TSHRMAPTLMNA
SCHEMBL7170671 0.89 ALDH1A1 (0.47) ALDH1A1CYP3A4TSHRMAPTLMNA
SCHEMBL5949786 0.81 ALDH1A1 (0.47) ALDH1A1CYP3A4TSHRMAPTLMNA
SCHEMBL7121793 0.80 GAA (0.46) ALDH1A1CYP3A4TSHRMAPTLMNA
SCHEMBL7784764 0.80 ALDH1A1 (0.42) ALDH1A1CYP3A4TSHRMAPTLMNA
SCHEMBL29493797 0.80 ALDH1A1 (0.42) ALDH1A1CYP3A4TSHRMAPTLMNA
SCHEMBL4594350 0.77 ALDH1A1 (0.48) ALDH1A1CYP3A4TSHRMAPTHPGD
SCHEMBL8653908 0.77 ALDH1A1 (0.50) ALDH1A1CYP3A4TSHRMAPTHPGD
SCHEMBL1192005 0.77 ALDH1A1 (0.50) ALDH1A1CYP3A4TSHRMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP disclosed
EP-0970100-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-01-12 EP disclosed
WO-1998035977-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1998-08-20 WO disclosed