SCHEMBL7115131

SCHEMBL7115131

[c]1c(-c2cc3ccccc3[nH]2)cc[nH]c2nnc1-2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.42
ESR1 P03372 3/20 0.40
ITK Q08881 4/20 0.39
CYP19A1 P11511 1/20 0.39
KDM4E B2RXH2 4/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
KMT2A Q03164 3/20 0.39
CASP3 P42574 2/20 0.39
SENP8 Q96LD8 2/20 0.39
SENP7 Q9BQF6 2/20 0.39
SENP6 Q9GZR1 2/20 0.39
CHEK1 O14757 1/20 0.39
KDR P35968 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689765 0.70 RAB9A (0.52) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL467441 0.69 RAB9A (0.50) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL2894778 0.69 ESR1 (0.51) RAB9ANPC1ESR1ITKCYP19A1
Benzene SCHEMBL28123406 0.68 RAB9A (0.53) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL29631691 0.68 RAB9A (0.74) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL374022 0.68 RAB9A (0.74) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL28399450 0.67 RAB9A (0.61) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL1781163 0.66 RAB9A (0.55) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL690118 0.66 CYP19A1 (0.53) RAB9ANPC1ESR1ITKCYP19A1
SCHEMBL7194943 0.65 KDR (0.56) RAB9ANPC1ESR1ITKCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030220400-A1 Enantiomerically pure basic arylcycloalkylhydroxycarboxylic esters, processes for their preparation and their use in medicaments Noe, Christian 2003-11-27 US disclosed
US-6307060-B1 ANTISPASMODIC AGENTS Noe, Christian 2001-10-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030220400-A1 Enantiomerically pure basic arylcycloalkylhydroxycarboxylic esters, processes for their preparation and their use in medicaments CYP2A13, CYP3A43, HCAR2 RAB9A 4658/4885NPC1 1409/4885ESR1 1163/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.