SCHEMBL7115446

SCHEMBL7115446

O=S(=O)(O)c1ccc(-c2c(-c3cccc(C(F)(F)F)c3)noc2C(F)F)cc1F

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.40
GPBAR1 Q8TDU6 1/20 0.36
MAPT P10636 3/20 0.35
GAA P10253 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MCOLN3 Q8TDD5 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
MAOB P27338 1/20 0.34
ELANE P08246 1/20 0.34
PTPN1 P18031 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
IP6K1 Q92551 1/20 0.34
IP6K3 Q96PC2 1/20 0.34
IP6K2 Q9UHH9 1/20 0.34
PTGS2 P35354 1/20 0.33
RORB Q92753 1/20 0.33
S1PR1 P21453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6723024 0.90 BRD4 (0.42) BRD4GPBAR1MAPTGAANPSR1
SCHEMBL6729567 0.90 BRD4 (0.42) BRD4GPBAR1MAPTGAANPSR1
SCHEMBL7112147 0.83 GABRG2 (0.35) MAOB
SCHEMBL7110955 0.82 MAPK14 (0.36) PTPN1PTGS2
SCHEMBL6732481 0.82 CA1 (0.41) BRD4GPBAR1MAPTGAANPSR1
SCHEMBL7108397 0.81 MAPK14 (0.38) NPSR1MCOLN3PTGS2
SCHEMBL6722729 0.79 PTGS2 (0.41) PTGS2
SCHEMBL6726764 0.79 PTGS2 (0.42) PTGS2
SCHEMBL6739355 0.79 BRD4 (0.39) BRD4GPBAR1MAPTGAANPSR1
SCHEMBL6719025 0.78 PTGS2 (0.43) BRD4GPBAR1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296971-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2003-04-02 EP disclosed
WO-2001081332-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2001-11-01 WO disclosed