SCHEMBL7116337

SCHEMBL7116337

O=C(O)c1ccn2c1-c1ccccc1CC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.41
SRD5A1 P18405 1/20 0.41
SRD5A2 P31213 1/20 0.41
KDM4E B2RXH2 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MTNR1A P48039 3/20 0.38
MTNR1B P49286 3/20 0.38
ALDH1A1 P00352 5/20 0.38
HPGD P15428 2/20 0.38
LMNA P02545 1/20 0.38
NOTUM Q6P988 1/20 0.38
PTAFR P25105 1/20 0.37
BCAT2 O15382 1/20 0.37
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36
SERPINE1 P05121 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1159572 0.89 MTNR1A (0.43) KDM4ENPC1RAB9AMAPTPKM
SCHEMBL10670409 0.76 KDM4E (0.39) L3MBTL1SRD5A1SRD5A2KDM4ENPC1
SCHEMBL28633869 0.76 MAPT (0.50) KDM4ENPC1RAB9AMAPTPKM
SCHEMBL1159362 0.73 KDM4E (0.41) L3MBTL1KDM4ENPC1RAB9AMAPT
SCHEMBL2780444 0.73 PDE10A (0.40) SRD5A1SRD5A2KDM4ENPC1RAB9A
SCHEMBL30712298 0.73 NPC1 (0.44) KDM4ENPC1RAB9AMAPTPKM
SCHEMBL29376705 0.71 KDM4E (0.56) L3MBTL1SRD5A1SRD5A2KDM4ENPC1
SCHEMBL16973636 0.71 KDM4E (0.56) L3MBTL1SRD5A1SRD5A2KDM4ENPC1
SCHEMBL9334779 0.69 TSHR (0.40) L3MBTL1SRD5A1SRD5A2KDM4ENPC1
SCHEMBL215395 0.67 SERPINE1 (0.39) L3MBTL1SRD5A1SRD5A2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003014115-A1 3-SUBSTITUTED PYRROLO (2.1-A) ISOQUINOLINE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2003-02-20 WO disclosed
WO-2003014117-A1 3-SUBSTITUTED PYRROLO[2.1-A]ISOQUINOLINE DERIVATIVES BAYER CORPORATION (US) 2003-02-20 WO disclosed