SCHEMBL7118397

SCHEMBL7118397

COC(=O)c1cccc(-c2cc3nccc(Cl)c3s2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
CES1 P23141 2/20 0.42
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MRGPRX4 Q96LA9 2/20 0.39
TYK2 P29597 2/20 0.38
MAPT P10636 3/20 0.38
CYP1A2 P05177 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 1/20 0.38
RECQL P46063 1/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5242363 0.80 NPC1 (0.42) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL5240149 0.80 MAOA (0.46) ALDH1A1RAB9AKDM4EHPGDL3MBTL1
SCHEMBL7123516 0.79 ERN1 (0.43) ALDH1A1NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL5241139 0.79 ALDH1A1 (0.37) ALDH1A1MRGPRX4TYK2ALOX15HTT
SCHEMBL7123648 0.78 GRM5 (0.41) NPC1RAB9AGRM5
SCHEMBL7126957 0.77 HTR2C (0.44) ALDH1A1NPC1RAB9AHPGDMAPT
SCHEMBL7125950 0.75 MCHR1 (0.35) NPC1RAB9ATYK2JAK2
SCHEMBL1460546 0.75 KDR (0.46) ALDH1A1HPGDMRGPRX4TYK2ALOX15
SCHEMBL29368150 0.75 KDR (0.46) ALDH1A1HPGDMRGPRX4TYK2ALOX15
SCHEMBL7123672 0.75 MCHR1 (0.41) RAB9AKDM4ETYK2SMN1; SMN2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030162795-A1 Thienopyrimidine and thienopyridine derivatives useful as anticancer agents PFIZER INC. 2003-08-28 US disclosed
US-6492383-B1 Thienopyrimidine and thienopyridine derivatives useful as anticancer agents PFIZER INC. 2002-12-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030162795-A1 Thienopyrimidine and thienopyridine derivatives useful as anticancer agents TYMP, DPYD, HPRT1 ALDH1A1 226/4885CES1 1254/4885NPC1 2221/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.