SCHEMBL7119177

SCHEMBL7119177

O=C1CN(CC2CCCCC2NC(=O)OCc2ccccc2)CC(Cc2ccc(F)cc2)N1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 16/20 0.48
CASP3 P42574 3/20 0.42
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
CYP2D6 P10635 1/20 0.41
DRD2 P14416 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3879488 1.00 CCR3 (0.48) CCR3CASP3CTSLCTSBCTSS
SCHEMBL3886795 0.95 CTSB (0.45) CCR3CASP3CTSLCTSBCTSS
SCHEMBL3886799 0.95 CTSB (0.45) CCR3CASP3CTSLCTSBCTSS
SCHEMBL3878046 0.83 HDAC6 (0.46) CCR3CASP3CTSLCTSBCTSS
SCHEMBL7112217 0.83 HDAC6 (0.46) CCR3CASP3CTSLCTSBCTSS
SCHEMBL3881417 0.83 CCR3 (0.43) CCR3CASP3CTSLCTSBCTSS
SCHEMBL13867601 0.80 CCR3 (0.43) CCR3CYP2D6DRD2SLC6A2HTR2A
SCHEMBL3881200 0.80 CCR3 (0.57) CCR3CYP2D6DRD2SLC6A2HTR2A
SCHEMBL3881197 0.80 CCR3 (0.57) CCR3CYP2D6DRD2SLC6A2HTR2A
SCHEMBL3881565 0.80 CCR3 (0.57) CCR3CYP2D6DRD2SLC6A2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003024401-A2 PIPERIZINONES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2003-03-27 WO disclosed