SCHEMBL7121835

SCHEMBL7121835

Cc1c(CC(N)=O)c(=O)oc2cccc(N)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.40
HSD17B10 Q99714 4/20 0.40
GAA P10253 2/20 0.40
CASP1 P29466 2/20 0.40
CASP7 P55210 2/20 0.40
RXFP1 Q9HBX9 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
TP53 P04637 2/20 0.40
ALDH1A1 P00352 6/20 0.40
HPGD P15428 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 1/20 0.40
NQO1 P15559 1/20 0.39
SLC26A3 P40879 4/20 0.39
MAPT P10636 1/20 0.38
GLA P06280 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2522181 0.89 TP53 (0.50) KDM4EHSD17B10PTGDR2TP53ALDH1A1
SCHEMBL29579782 0.79 PSMB8 (0.45) KDM4EHSD17B10GAACASP1CASP7
SCHEMBL6578104 0.75 CA12 (0.49) KDM4EHSD17B10GAAALDH1A1HPGD
SCHEMBL3994327 0.73 SRC (0.64) KDM4EHSD17B10GAACASP1CASP7
SCHEMBL5085076 0.72 TP53 (0.51) KDM4EHSD17B10GAACASP1CASP7
SCHEMBL27593866 0.69 EDNRA (0.62) KDM4EHSD17B10ALDH1A1HPGDMAPT
SCHEMBL21665556 0.67 CYP3A4 (0.48) KDM4EHSD17B10GAACASP1CASP7
SCHEMBL10794643 0.67 MAPT (0.52) KDM4EHSD17B10GAACASP1CASP7
SCHEMBL3609409 0.67 RAB9A (0.72) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL4100411 0.66 CYP3A4 (0.48) KDM4EHSD17B10GAANPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003029823-A1 COMBINATORIAL PROTEASE SUBSTRATE LIBRARIES IRM LLC (BM) 2003-04-10 WO claimed
US-20030059847-A1 Combinatorial protease substrate libraries IRM, LLC (BM) 2003-03-27 US claimed