SCHEMBL7123726

SCHEMBL7123726

O=C(O)N1CCN(c2cccc(CS(=O)(=O)C=C3CN(C(c4ccc(Cl)cc4)c4ccc(Cl)cc4)C3)c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
LMNA P02545 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
RECQL P46063 1/20 0.40
CACNA2D1 P54289 4/20 0.40
CACNB1 Q02641 4/20 0.40
CACNA1B Q00975 3/20 0.40
CACNA1C Q13936 3/20 0.40
MAPT P10636 3/20 0.40
GAA P10253 2/20 0.40
CACNA1G O43497 2/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GRM5 P41594 1/20 0.40
GFER P55789 1/20 0.40
ATM Q13315 1/20 0.40
CACNA1A O00555 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7127512 0.92 TP53 (0.39) TP53LMNANPSR1TSHRMAPK1
SCHEMBL6011709 0.92 CYP3A4 (0.43) TP53LMNANPSR1TSHRMAPK1
SCHEMBL6011624 0.90 CACNA1G (0.42) CACNA2D1CACNB1CACNA1BCACNA1CMAPT
SCHEMBL6011378 0.89 SMN1; SMN2 (0.42) TP53LMNANPSR1TSHRMAPK1
SCHEMBL6011475 0.89 LMNA (0.44) TP53LMNANPSR1TSHRMAPK1
SCHEMBL6011563 0.89 HRH3 (0.42) TP53LMNANPSR1TSHRMAPK1
SCHEMBL6011760 0.88 KMT2A (0.42) LMNACACNA2D1CACNB1CACNA1BCACNA1C
SCHEMBL6011681 0.88 SMN1; SMN2 (0.43) TP53LMNANPSR1MAPK1CACNA2D1
SCHEMBL6011783 0.87 HTT (0.44) TP53NPSR1MAPTHTTMEN1
SCHEMBL6011554 0.87 MAPT (0.43) LMNANPSR1TSHRMAPK1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112251-B1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM AVENTIS PHARMA SA (FR) 2003-05-07 EP claimed