Monomethyl Fumarate

Monomethyl Fumarate

SCHEMBL7123923

C=C(C)OC(=C)C.COC(=O)/C=C\C(=O)O

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Monomethyl Fumarate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.54
HCAR2 Q8TDS4 9/20 0.71
ALDH1A1 P00352 4/20 0.55
TDP1 Q9NUW8 2/20 0.55
KDM4E B2RXH2 1/20 0.55
MAPT P10636 1/20 0.55
NFE2L2 Q16236 1/20 0.54
HSD17B10 Q99714 2/20 0.52
ALOX15 P16050 1/20 0.52
RECQL P46063 1/20 0.52
TSHR P16473 3/20 0.38
TP53 P04637 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
EGLN3 Q9H6Z9 1/20 0.38
GFPT1 Q06210 1/20 0.36
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Monomethyl Fumarate SCHEMBL7764250 0.89 HCAR2 (0.81) HCAR2ALDH1A1TDP1KDM4EMAPT
Fumaric Acid SCHEMBL3701419 0.87 HSD17B10 (0.52) HCAR2ALDH1A1TDP1KDM4EMAPT
Maleic Acid SCHEMBL251369 0.87 HSD17B10 (0.52) HCAR2ALDH1A1TDP1KDM4EMAPT
SCHEMBL4168638 0.85 HCAR2 (0.52) HCAR2ALDH1A1TDP1KDM4EMAPT
SCHEMBL1014778 0.85 HCAR2 (0.52) HCAR2ALDH1A1TDP1KDM4EMAPT
Monomethyl Fumarate SCHEMBL5607806 0.84 HCAR2 (0.90) HCAR2ALDH1A1TDP1KDM4EMAPT
Fumaric Acid SCHEMBL9248586 0.84 HSD17B10 (0.50) HCAR2ALDH1A1TDP1KDM4EMAPT
Maleic Acid SCHEMBL4507841 0.84 HSD17B10 (0.50) HCAR2ALDH1A1TDP1KDM4EMAPT
Monomethyl Fumarate SCHEMBL5607800 0.84 HCAR2 (0.90) HCAR2ALDH1A1TDP1KDM4EMAPT
Monomethyl Fumarate SCHEMBL25280962 0.84 HCAR2 (1.00) HCAR2ALDH1A1TDP1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030139502-A1 Cosmetic compositions comprising a cationic polymer/anionic surfactant mixture and use of said mixture as conditioning agent RHODIA CHIMIE (FR) 2003-07-24 US disclosed
US-4265778-A FATTY ACID SALT, INTERPOLYMER OF A MALEIC ANHYDRIDE OR ACID AND A VINYL LACTAM OR VINYL ETHER OR ESTER COLGATE-PALMOLIVE COMPANY (US) 1981-05-05 US disclosed