SCHEMBL7126729

SCHEMBL7126729

O=C(O)NN1CCc2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
HPGD P15428 2/20 0.51
SMN1; SMN2 Q16637 6/20 0.51
NPC1 O15118 5/20 0.51
RAB9A P51151 5/20 0.51
NFKB1 P19838 3/20 0.51
NFKB2 Q00653 3/20 0.51
RELA Q04206 3/20 0.51
PKM P14618 2/20 0.51
TP53 P04637 2/20 0.51
NOTUM Q6P988 2/20 0.50
MAPT P10636 3/20 0.49
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
TSHR P16473 2/20 0.49
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29985725 1.00 ALDH1A1 (0.51) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL27745558 0.90 SMN1; SMN2 (0.56) ALDH1A1HPGDSMN1; SMN2NOTUMMAPT
Hydrochloric Acid SCHEMBL1859868 0.88 SMN1; SMN2 (0.54) ALDH1A1HPGDSMN1; SMN2NOTUMMAPT
SCHEMBL5120536 0.86 NOTUM (0.50) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL31488059 0.84 NOTUM (0.57) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL28650278 0.78 MAPT (0.53) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL307373 0.78 TSHR (0.45) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL7045087 0.78 NPC1 (0.61) ALDH1A1SMN1; SMN2NPC1RAB9ANFKB1
SCHEMBL4984050 0.77 SIGMAR1 (0.51) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL11348161 0.77 SIGMAR1 (0.43) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100334076-C Indoline derivatives and their use as 5-HT2Use of receptor ligands HOFFMANN LA ROCHE CO LTD (CH) 2007-08-29 CN disclosed
EP-1328515-A1 INDOLINE DERIVATIVES AND THEIR USE AS 5-HT2 RECEPTOR LIGANDS F. Hoffmann-La Roche AG (CH) 2003-07-23 EP disclosed
WO-2002044152-A1 INDOLINE DERIVATIVES AND THEIR USE AS 5-HT2 RECEPTOR LIGANDS F. HOFFMANN-LA ROCHE AG (CH) 2002-06-06 WO disclosed