SCHEMBL7126736

SCHEMBL7126736

COc1ccc(Cc2cnc(N)nc2N)cc1I

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.78
HTT P42858 1/20 0.78
NTRK1 P04629 1/20 0.65
CSF1R P07333 1/20 0.65
NTRK3 Q16288 1/20 0.65
NTRK2 Q16620 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diaveridine SCHEMBL93896 0.88 DHFR (1.00) DHFRHTTNTRK1CSF1RNTRK3
Diaveridine SCHEMBL29527560 0.88 DHFR (1.00) DHFRHTTNTRK1CSF1RNTRK3
SCHEMBL9657245 0.84 DHFR (0.78) DHFRHTTNTRK1CSF1RNTRK3
SCHEMBL9830386 0.84 DHFR (0.82) DHFRHTTNTRK1CSF1RNTRK3
SCHEMBL5943361 0.83 DHFR (0.82) DHFR
Hydrochloric Acid SCHEMBL11385904 0.83 DHFR (0.76) DHFRHTTNTRK1CSF1RNTRK3
SCHEMBL10488908 0.83 DHFR (0.85) DHFRHTTNTRK1CSF1RNTRK3
SCHEMBL11596783 0.82 DHFR (0.77) DHFRHTT
SCHEMBL2680692 0.82 DHFR (0.68) DHFRHTT
SCHEMBL9654048 0.82 DHFR (0.78) DHFRHTTNTRK1CSF1RNTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1136198-C Novel benzyl pyrimidines ��������ҩ�ɷ����޹�˾ 2004-01-28 CN disclosed
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
CN-1166831-A Novel benzyl pyrimidines HOFFMANN LA ROCHE (CH) 1997-12-03 CN disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed