SCHEMBL7126899

SCHEMBL7126899

NCCOc1cccc2cc(Br)ccc12

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 7/20 0.65
KDM4E B2RXH2 3/20 0.47
KCNA3 P22001 1/20 0.41
HTR1D P28221 1/20 0.41
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
SLC6A4 P31645 2/20 0.40
HRH1 P35367 1/20 0.40
MAPT P10636 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
NCF1 P14598 2/20 0.39
NR2E1 Q9Y466 1/20 0.39
ITK Q08881 1/20 0.39
CYBB P04839 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17919856 0.83 HTR1B (0.51) HTR1BKCNA3HTR1DSLC6A4HRH1
SCHEMBL15565685 0.80 HTR1B (0.49) HTR1BKCNA3HTR1DSLC6A4HRH1
SCHEMBL9523932 0.79 HTR1B (1.00) HTR1BKDM4EKCNA3HTR1DSLC6A4
SCHEMBL30825865 0.79 HTR1B (1.00) HTR1BKDM4EKCNA3HTR1DSLC6A4
Hydrochloric Acid SCHEMBL12465902 0.77 NCEH1 (0.49) HTR1BKDM4EMAPTLMNAMAPK1
SCHEMBL7415980 0.76 ERN1 (0.40) HTR1BKDM4EKCNA3HTR1D
SCHEMBL17913768 0.76 MAOB (0.53) SLC6A4MAPTMAPK1RAB9A
SCHEMBL29576746 0.76 MAOB (0.53) SLC6A4MAPTMAPK1RAB9A
SCHEMBL7415972 0.76 DAO (0.39) HTR1BKDM4EKCNA3HTR1DSLC6A4
SCHEMBL24801284 0.74 CYP2A6 (0.43) KDM4ESLC6A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030114448-A1 Inhibitors of factor Xa MILLENNIUM PHARMACEUTICALS, INC. 2003-06-19 US disclosed
WO-2002096873-A1 ISOINDOLE AND ISOQUINOLINE DERIVATIVES AS INHIBITORS OF FACTOR XA MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-12-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114448-A1 Inhibitors of factor Xa SERPINC1, F11, TFPI HTR1B 3888/4885KDM4E 3179/4885KCNA3 2630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.