SCHEMBL7415972

SCHEMBL7415972

O=[C]COc1cccc2cc(Br)ccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.39
MCL1 Q07820 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTR1B P28222 3/20 0.36
HTR1D P28221 1/20 0.36
CYP2A6 P11509 2/20 0.36
SLC6A4 P31645 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HRH1 P35367 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
CYP3A4 P08684 1/20 0.35
APAF1 O14727 1/20 0.35
TDP2 O95551 1/20 0.35
SLC6A2 P23975 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2121728 0.80 KDM4E (0.56) KDM4EALDH1A1HPGDTDP1HTR1B
SCHEMBL7415980 0.78 ERN1 (0.40) DAOMCL1KDM4EALDH1A1HPGD
SCHEMBL7126899 0.76 HTR1B (0.65) KDM4EHTR1BHTR1DSLC6A4HRH1
SCHEMBL17919856 0.75 HTR1B (0.51) HTR1BHTR1DSLC6A4HRH1CYP1A2
SCHEMBL17913768 0.75 MAOB (0.53) ALDH1A1TDP1SLC6A4MEN1KMT2A
SCHEMBL29576746 0.75 MAOB (0.53) ALDH1A1TDP1SLC6A4MEN1KMT2A
SCHEMBL5804242 0.73 MAPK1 (0.52) ALDH1A1HPGDTDP1HTR1BMEN1
SCHEMBL24801284 0.73 CYP2A6 (0.43) DAOKDM4EALDH1A1HPGDTDP1
SCHEMBL6312903 0.73 KDM4E (0.51) KDM4EALDH1A1HPGDCYP2A6MEN1
SCHEMBL15565685 0.73 HTR1B (0.49) HTR1BHTR1DSLC6A4HRH1KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013066-A1 CYCLIC AMIDES OF 3-AMINO-2-HYDROXY-CARBOXYLIC ACIDS AS HIV-PROTEASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1993-07-08 WO disclosed