SCHEMBL7127951

SCHEMBL7127951

CCCCCNC(=O)C(Cc1ccc(N)c(I)c1)NC(=O)[CH]Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47
PTPN1 P18031 7/20 0.45
CHRND Q07001 5/20 0.44
CHRNA1 P02708 3/20 0.44
CHRNG P07510 3/20 0.44
CHRNB1 P11230 3/20 0.44
PLG P00747 2/20 0.44
PRSS1 P07477 2/20 0.44
PRSS2 P07478 2/20 0.44
PRSS3 P35030 2/20 0.44
KLKB1 P03952 1/20 0.44
GRIA1 P42261 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPRA P18433 1/20 0.43
TLR2 O60603 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7127958 0.85 PTPN1 (0.60) CHRNB2CHRNB4CHRNA3CHRNA4PTPN1
SCHEMBL7571008 0.80 PTPN1 (0.58) CHRNB2CHRNB4CHRNA3CHRNA4PTPN1
SCHEMBL7569835 0.80 PTPN1 (0.67) PTPN1PTPRA
SCHEMBL7066343 0.78 PTPN1 (0.57) PTPN1PLGPRSS1PRSS2PRSS3
SCHEMBL7065637 0.77 PTPN1 (0.51) PTPN1CHRNDCHRNA1CHRNGCHRNB1
SCHEMBL7571014 0.77 PTPN1 (0.52) CHRNB2CHRNB4CHRNA3CHRNA4PTPN1
SCHEMBL7065286 0.77 DPP7 (0.49) GRIA1
SCHEMBL10545669 0.72 CHRNB2 (0.67) CHRNB2CHRNB4CHRNA3CHRNA4CHRND
SCHEMBL988166 0.72 CHRNB2 (0.77) CHRNB2CHRNB4CHRNA3CHRNA4CHRND
SCHEMBL5933899 0.71 EGFR (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313696-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2003-05-28 EP disclosed
WO-2002018323-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2002-03-07 WO disclosed