SCHEMBL7127958

SCHEMBL7127958

CCCCCNC(=O)C(Cc1ccc(N)c(I)c1)NC(=O)CCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.60
GRIA1 P42261 2/20 0.57
CHRNB2 P17787 2/20 0.56
CHRNB4 P30926 2/20 0.56
CHRNA3 P32297 2/20 0.56
CHRNA4 P43681 2/20 0.56
HPGD P15428 1/20 0.54
CHRND Q07001 6/20 0.52
CHRNA1 P02708 2/20 0.52
CHRNG P07510 2/20 0.52
CHRNB1 P11230 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7571008 0.87 PTPN1 (0.58) PTPN1GRIA1CHRNB2CHRNB4CHRNA3
SCHEMBL7127951 0.85 CHRNB2 (0.47) PTPN1GRIA1CHRNB2CHRNB4CHRNA3
SCHEMBL7569835 0.82 PTPN1 (0.67) PTPN1
SCHEMBL988166 0.80 CHRNB2 (0.77) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7571014 0.80 PTPN1 (0.52) PTPN1GRIA1CHRNB2CHRNB4CHRNA3
SCHEMBL7066343 0.80 PTPN1 (0.57) PTPN1GRIA1
SCHEMBL12324830 0.79 CHRNB2 (0.69) PTPN1GRIA1CHRNB2CHRNB4CHRNA3
SCHEMBL6438848 0.79 CHRNB2 (0.69) PTPN1GRIA1CHRNB2CHRNB4CHRNA3
SCHEMBL16247369 0.79 CHRNB2 (0.69) PTPN1GRIA1CHRNB2CHRNB4CHRNA3
SCHEMBL9519035 0.79 CHRNB2 (0.69) PTPN1GRIA1CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313696-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2003-05-28 EP disclosed
WO-2002018323-A2 AMINO(OXO)ACETIC ACID PROTEIN TYROSINE PHOSPHATASE INHIBITORS ABBOTT LABORATORIES (US) 2002-03-07 WO disclosed