Lonidamine

Lonidamine

SCHEMBL7134

O=C(O)c1nn(Cc2ccc(Cl)cc2Cl)c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 1.00
CYP3A4 P08684 2/20 1.00
CYP2C9 P11712 2/20 1.00
CYP2D6 P10635 1/20 1.00
TSHR P16473 1/20 1.00
PMP22 Q01453 1/20 1.00
HIF1A Q16665 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
PTGER4 P35408 4/20 0.52
SLC9A1 P19634 1/20 0.51
LMNA P02545 4/20 0.51
ALDH1A1 P00352 3/20 0.51
MAPT P10636 2/20 0.51
ALOX12 P18054 1/20 0.51
NPC1 O15118 1/20 0.51
MCL1 Q07820 1/20 0.47
KDM4E B2RXH2 1/20 0.46
GLA P06280 1/20 0.46
HPGD P15428 1/20 0.46
PTGER1 P34995 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lonidamine SCHEMBL29351122 1.00 CYP1A2 (1.00) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
Lonidamine SCHEMBL29350056 1.00 CYP1A2 (1.00) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
Lonidamine SCHEMBL28075715 0.93 CYP1A2 (0.87) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
Lonidamine SCHEMBL28086501 0.92 CYP1A2 (0.85) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
Lonidamine SCHEMBL5483035 0.91 CYP1A2 (0.83) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
SCHEMBL31566279 0.90 CYP1A2 (0.82) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
SCHEMBL14584151 0.90 CYP1A2 (0.82) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
SCHEMBL21121979 0.90 CYP1A2 (0.82) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
SCHEMBL30949037 0.90 CYP1A2 (0.81) CYP1A2CYP3A4CYP2C9CYP2D6TSHR
SCHEMBL1051466 0.90 CYP1A2 (0.81) CYP1A2CYP3A4CYP2C9CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 31492 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122080068-A Mitochondria-targeted lonidamine and cinnamaldehyde coupled prodrug as well as preparation method and application thereof 2026-05-26 CN claimed
CN-122075505-A Ternary nanoparticle and preparation method and application thereof 2026-05-26 CN claimed
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF SYSTIMMUNE INC (US) 2026-05-21 US claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-20260109699-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2026-04-23 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-3515892-B1 COMPOUNDS AND METHODS FOR IDO AND TDO MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC (US) 2026-04-15 EP claimed
US-20260085100-A1 METHODS OF ANTIGEN PRODUCTION THE WISTAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2026-03-26 US claimed
US-20260085061-A1 PHTHALAZINE DERIVATIVES AS PYRUVATE KINASE MODULATORS SITRYX THERAPEUTICS LIMITED (GB) 2026-03-26 US claimed
EP-0642799-A1 Improved prodrugs for enzyme mediated activation BEHRINGWERKE Aktiengesellschaft (DE) 1995-03-15 EP claimed
EP-0393575-B1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent SEARLE & CO (US) 1994-03-16 EP claimed
US-5260327-A Methods for inhibiting the proliferation of brain and hepatic metastases by using lonidamine SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1993-11-09 US claimed
EP-0172721-B1 USE OF PHLORIZIN OR ITS DERIVATIVES IN COMBINATION WITH A CHEMOTHERAPEUTIC AGENT FOR THE TREATMENT OF CANCER Leveen, Harry H. (US) 1993-03-03 EP claimed
EP-0393575-A1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent G.D. Searle & Co. (US) 1990-10-24 EP claimed
US-4840939-A Treatment of cancer with phlorizin and its derivatives LEVEEN HARRY H (US) 1989-06-20 US claimed
EP-0291151-A1 Compositions comprising phlorizin derivatives for treatment of cancer Leveen, Harry H. (US) 1988-11-17 EP claimed
US-4684627-A Treatment of cancer with phlorizin and its derivatives MEDICINAL DEVELOPMENTS,INC. 1987-08-04 US claimed
EP-0172721-A2 Use of phlorizin or its derivatives in combination with a chemotherapeutic agent for the treatment of cancer Leveen, Harry H. (US) 1986-02-26 EP claimed
US-4282237-A Method with substituted 1-benzyl-1H-indazole-3-carboxylic acids for interrupting pregnancy in mammals AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A. (IT) 1981-08-04 US claimed