SCHEMBL7135262

SCHEMBL7135262

CCOC(=O)/C=C/c1cc2ccccc2n1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.45
DPP4 P27487 1/20 0.45
ALB P02768 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CYP3A4 P08684 2/20 0.44
CCNC P24863 2/20 0.44
CDK8 P49336 2/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MCL1 Q07820 1/20 0.43
PTGS2 P35354 1/20 0.43
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7135266 1.00 TTR (0.45) TTRDPP4ALBCA12CA1
SCHEMBL6364609 0.85 ALB (0.47) TTRALBCA12CA1CA2
SCHEMBL6364611 0.85 ALB (0.47) TTRALBCA12CA1CA2
SCHEMBL12355545 0.82 MEN1 (0.48) TTRDPP4CA12CA1CA2
SCHEMBL3204531 0.81 ALB (0.49) ALBNPC1RAB9AMCL1GRIN2D
SCHEMBL3204520 0.81 ALB (0.49) ALBNPC1RAB9AMCL1GRIN2D
SCHEMBL6364102 0.81 LMNA (0.45) TTRDPP4CA12CA1CA2
SCHEMBL6364105 0.81 LMNA (0.45) TTRDPP4CA12CA1CA2
SCHEMBL29247884 0.80 GRIN2D (0.51) ALBNPC1RAB9AMCL1GRIN2D
SCHEMBL7326486 0.80 MCL1 (0.54) ALBNPC1RAB9AMCL1GRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596738-B1 Inhibiting activity to adenosine deaminase (hereinafter described as ADA) An adenosine deaminase inhibiting agent comprising a compound of the formula (I): FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-22 US disclosed
EP-0392663-A1 Carboline derivative as a 5-HT3 receptor antagonist ONO PHARMACEUTICAL CO., LTD. (JP) 1990-10-17 EP disclosed