SCHEMBL7140696

SCHEMBL7140696

COc1cc(OC)cc(S(=O)(=O)c2ccc([N+](=O)[O-])c(C)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.48
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
VCAM1 P19320 1/20 0.44
PKM P14618 1/20 0.43
POLB P06746 2/20 0.43
MCOLN3 Q8TDD5 1/20 0.43
MAPT P10636 3/20 0.43
TSHR P16473 2/20 0.42
RAPGEF4 Q8WZA2 1/20 0.41
MAPK1 P28482 3/20 0.40
ALDH1A1 P00352 2/20 0.40
S1PR4 O95977 1/20 0.40
S1PR1 P21453 1/20 0.40
RAB9A P51151 1/20 0.40
GFER P55789 1/20 0.40
PAX8 Q06710 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144573 0.78 PTGS1 (0.62) PTGS1PTGS2PKMPOLBALDH1A1
SCHEMBL2478404 0.78 KMT2A (0.56) VCAM1POLBMAPTTSHRMAPK1
SCHEMBL30382526 0.77 ALDH1A1 (0.57) POLBMCOLN3MAPTTSHRMAPK1
SCHEMBL1897174 0.77 ALDH1A1 (0.57) POLBMCOLN3MAPTTSHRMAPK1
SCHEMBL7536269 0.77 PKM (0.61) VCAM1PKMPOLBMCOLN3MAPT
SCHEMBL7136138 0.77 PKM (0.47) CYP19A1PTGS1PTGS2PKMPOLB
SCHEMBL6516381 0.74 MAPT (0.53) PKMMCOLN3MAPTTSHRALDH1A1
SCHEMBL27470882 0.74 PKM (0.47) CYP19A1PTGS2PKMPOLBMAPT
SCHEMBL7142272 0.73 MAPT (0.43) CYP19A1PTGS1PTGS2PKMMAPT
SCHEMBL1828638 0.73 MAPT (0.51) VCAM1MCOLN3MAPTTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0930302-B1 Benzosulfone derivatives HOFFMANN LA ROCHE (CH) 2003-04-02 EP disclosed
US-5990105-A POSSESS A SELECTIVE AFFINITY TO 5HT-6 RECEPTORS; TREATING OR PREVENTING PSYCHOSES, SCHIZOPHRENIA, MANIC DEPRESSIONS, DEPRESSIONS, NEUROLOGICAL DISORDERS, PARKINSON'S, AMYOTROPHIC LATERAL SCLEROSIS, ALZHEIMER'S AND HUNTINGTON'S DISEASE HOFFMANN-LA ROCHE INC. (US) 1999-11-23 US disclosed
EP-0930302-A2 Benzosulfone derivatives F.HOFFMANN-LA ROCHE AG (CH) 1999-07-21 EP disclosed