SCHEMBL7140812

SCHEMBL7140812

CO/C=C(/C(=O)O)c1ccccc1/C=C/C=C/c1sccc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.36
NPC1 O15118 5/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
MAPT P10636 7/20 0.33
ALDH1A1 P00352 6/20 0.33
KMT2A Q03164 5/20 0.33
MEN1 O00255 4/20 0.33
HPGD P15428 3/20 0.33
KDM4E B2RXH2 1/20 0.33
PSMD14 O00487 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
AR P10275 1/20 0.33
MAOB P27338 1/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GAA P10253 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7140815 1.00 RAB9A (0.36) RAB9ANPC1SMN1; SMN2MAPTALDH1A1
SCHEMBL7139094 0.80 MAOB (0.42) ALDH1A1KMT2AMEN1TDP1AR
SCHEMBL7139096 0.80 MAOB (0.42) ALDH1A1KMT2AMEN1TDP1AR
SCHEMBL7137664 0.79 SMN1; SMN2 (0.44) RAB9ANPC1SMN1; SMN2MAPTALDH1A1
SCHEMBL7137656 0.79 SMN1; SMN2 (0.44) RAB9ANPC1SMN1; SMN2MAPTALDH1A1
SCHEMBL7140256 0.78 LY96 (0.47) RAB9ANPC1MAPTALDH1A1KMT2A
SCHEMBL7140258 0.78 LY96 (0.47) RAB9ANPC1MAPTALDH1A1KMT2A
SCHEMBL7142506 0.78 ALDH1A1 (0.40) RAB9ANPC1SMN1; SMN2MAPTALDH1A1
SCHEMBL7142510 0.78 ALDH1A1 (0.40) RAB9ANPC1SMN1; SMN2MAPTALDH1A1
SCHEMBL7141735 0.77 MAPT (0.43) RAB9ANPC1MAPTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996439-B1 BETA-ALKOXYACRYLATES AGAINST MALARIA HOFFMANN LA ROCHE (CH) 2003-01-08 EP disclosed
US-6084120-A ACTIVE AGAINST CHLOROQUINE-SENSITIVE PATIENTS AND AGAINST CHLOROQUINE-RESISTANT MALARIA PATHOGENS; PROPHYLAXIS AND TREATMENT; E.G., A 3 METHOXY-2-(2-(4-PHENYLBUTA-1,3-DIEN-1-YL)PHENYL)ACRYLIC ACID HOFFMANN-LA ROCHE INC. (US) 2000-07-04 US disclosed