SCHEMBL7140970

SCHEMBL7140970

c1ccc(Cc2ccc(OCCN3CCCC3)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 15/20 1.00
PSMB1 P20618 1/20 0.84
PSMB5 P28074 1/20 0.84
PSMB2 P49721 1/20 0.84
HRH3 Q9Y5N1 2/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141103 0.98 LTA4H (1.00) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL7133844 0.98 LTA4H (1.00) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL7142387 0.92 HRH3 (0.97) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL8640984 0.91 HRH3 (0.89) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL8637452 0.91 HRH3 (1.00) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL7134882 0.90 LTA4H (1.00) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL7398931 0.88 HRH3 (0.89) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL8642188 0.88 LTA4H (0.78) LTA4HPSMB1PSMB5PSMB2HRH3
SCHEMBL2476820 0.87 LTA4H (1.00) LTA4HHRH3
Hydrochloric Acid SCHEMBL7397621 0.87 HRH3 (0.86) LTA4HPSMB1PSMB5PSMB2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220054429-A1 COMPOSITIONS COMPRISING CANNABIDIOL AND SECOND THERAPEUTIC AGENTS FOR THE TREATMENT OF CANCER AKOS BIOSCIENCES, INC. 2022-02-24 US claimed
US-20180311182-A1 COMPOSITIONS COMPRISING CANNABIDIOL AND SECOND THERAPEUTIC AGENTS FOR THE TREATMENT OF CANCER AKOS BIOSCIENCES, INC. 2018-11-01 US claimed
WO-2025242860-A2 PHYTOSTEROL DERIVATIVES, AND COMPOSITIONS COMPRISING THE SAME, FOR USE AS MEDICAMENTS Institut National de la Santé et de la Recherche Médicale (FR) 2025-11-27 WO disclosed
EP-4646421-A1 FLUORO-OXYSTEROLS POSITRON EMISSION TOMOGRAPHY (PET) RADIOTRACERS Institut National de la Santé et de la Recherche Médicale (FR) 2025-11-12 EP disclosed
WO-2024146880-A1 FLUORO-OXYSTEROLS POSITRON EMISSION TOMOGRAPHY (PET) RADIOTRACERS Institut National de la Santé et de la Recherche Médicale (FR) 2024-07-11 WO disclosed
EP-3097904-B1 DEPIGMENTING AGENTS TO LIGHTEN THE SKIN AFFICHEM (FR) 2019-08-14 EP disclosed
WO-2016193220-A1 SKIN PIGMENTATION MODIFIERS TO DARKEN OR LIGHTEN THE SKIN AFFICHEM (FR) 2016-12-08 WO disclosed
EP-3097904-A1 DEPIGMENTING AGENTS TO LIGHTEN THE SKIN Affichem (FR) 2016-11-30 EP disclosed
US-6506876-B1 LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. 2003-01-14 US disclosed
EP-0804427-B1 LTA4 HYDROLASE INHIBITORS SEARLE & CO (US) 2002-09-18 EP disclosed
EP-1221441-A2 LTA4 Hydrolase inhibitors G.D. SEARLE & CO. (US) 2002-07-10 EP disclosed
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed
EP-0804427-A1 LTA4 HYDROLASE INHIBITORS G.D. SEARLE & CO. (US) 1997-11-05 EP disclosed
EP-0786992-A2 LTA 4? HYDROLASE INHIBITOR PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE G.D. SEARLE & CO. (US) 1997-08-06 EP disclosed
US-5585492-A USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASES WHICH ARE MEDIATED BY LTB4 PRODUCTION, SUCH AS PSORIASIS, ULCERATIVE COLITIS, IRRITABLE BOWEL DISEASE AND ASTHMA G. D. SEARLE & CO. (US) 1996-12-17 US disclosed
WO-1996010999-A2 LTA4 HYDROLASE INHIBITOR PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE G.D. SEARLE & CO. (US) 1996-04-18 WO disclosed
WO-1996011192-A1 LTA4 HYDROLASE INHIBITORS G.D. SEARLE & CO. (US) 1996-04-18 WO disclosed