SCHEMBL7141244

SCHEMBL7141244

C#CCC(CC#C)C(=O)C(CC#C)CC#C

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.48
GRIK2 Q13002 2/20 0.48
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL379205 0.79 GRIK1 (0.64) GRIK1GRIK2
SCHEMBL8945452 0.77 GRIK1 (0.45) GRIK1GRIK2
SCHEMBL7200824 0.77 GRIK1 (0.50) GRIK1GRIK2
SCHEMBL8847145 0.73 GRIK1 (0.52) GRIK1GRIK2
SCHEMBL6870462 0.73
SCHEMBL9861585 0.73 GRIK1 (0.42) GRIK1GRIK2ALDH1A1
SCHEMBL19483357 0.71 GRIK1 (0.37) GRIK1GRIK2
SCHEMBL19483387 0.71 GRIK1 (0.37) GRIK1GRIK2
SCHEMBL7854706 0.71 CA1 (0.42) GRIK1GRIK2
SCHEMBL3104177 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6521604-B1 1,2-dicarba-closo-dodecarborane containing organic residue; reacting a decaborane with an acetylene; treating tumors DEUTCHES KREBSFORSCHUNGSZENTRUM (DE) 2003-02-18 US disclosed
EP-1051421-B1 COMPOUNDS CONTAINING BORON FOR ELECTRON MICROSCOPY AND FOR BORON NEUTRON-CAPTURE THERAPY DEUTSCHES KREBSFORSCH (DE) 2002-12-11 EP disclosed