SCHEMBL7141364

SCHEMBL7141364

c1cncc(NN2CCNCC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.47
CHRNA4 P43681 2/20 0.47
ADRA2A P08913 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
ROCK1 Q13464 1/20 0.43
ALDH1A1 P00352 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KCNA5 P22460 1/20 0.40
KCNH2 Q12809 1/20 0.40
POLB P06746 1/20 0.40
KMT2A Q03164 1/20 0.40
NAMPT P43490 2/20 0.39
GBA1 P04062 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7096492 0.84 CHRNB2 (0.44) CHRNB2CHRNA4ADRA2AADRA2BADRA2C
SCHEMBL6352342 0.82 LMNA (0.44) CHRNB2CHRNA4ALDH1A1POLBKMT2A
SCHEMBL7098715 0.82 LMNA (0.44) CHRNB2CHRNA4ALDH1A1POLBKMT2A
SCHEMBL2478525 0.79 SMN1; SMN2 (0.45) ALDH1A1KMT2ACYP3A4
SCHEMBL644787 0.77 POLB (0.49) ALDH1A1POLBKMT2ACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL6017637 0.77 ADRB2 (0.35) CHRNB2CHRNA4ROCK1ALDH1A1POLB
SCHEMBL1758868 0.73 POLB (0.66) MKNK1MKNK2POLBCYP1A2CYP2D6
SCHEMBL30791537 0.73 POLB (0.66) MKNK1MKNK2POLBCYP1A2CYP2D6
SCHEMBL28211335 0.73 RYR2 (0.50) CHRNB2CHRNA4ADRA2AADRA2BROCK1
SCHEMBL27915904 0.72 RPS6KA3 (0.39) CHRNB2CHRNA4ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289982-A1 BIOISOSTERIC BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2003-03-12 EP disclosed
WO-2001096327-A1 BIOISOSTERIC BENZAMIDE DERIVATIVES AND THEIR USE AS APoB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2001-12-20 WO disclosed