SCHEMBL7141863

SCHEMBL7141863

O=c1[nH]cc(OCCCC(F)(F)F)c2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.41
CYP2D6 P10635 1/20 0.40
PARP1 P09874 4/20 0.39
KDM4E B2RXH2 1/20 0.38
ROCK2 O75116 1/20 0.36
TNKS O95271 1/20 0.36
ROCK1 Q13464 1/20 0.36
PARP14 Q460N5 1/20 0.36
PARP10 Q53GL7 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
PARP3 Q9Y6F1 1/20 0.36
SCN8A Q9UQD0 4/20 0.36
SCN10A Q9Y5Y9 4/20 0.36
APP P05067 1/20 0.35
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KCNA3 P22001 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
GPR84 Q9NQS5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10989071 0.72 HTR1D (0.44) CYP2D6PARP1KDM4EKMT2AHSD17B10
SCHEMBL4451982 0.71 HRH3 (0.57) CYP2D6PARP1KDM4EKMT2A
SCHEMBL28043247 0.70 HTR1B (0.62) KMT2AKCNA3
SCHEMBL1536514 0.69 PARP1 (0.50) PARP1KDM4EKMT2AHSD17B10
SCHEMBL29531776 0.68 NCF1 (0.44) KCNA3
SCHEMBL7141860 0.68 PARP1 (0.36) PARP1KDM4EROCK2TNKSROCK1
SCHEMBL10608226 0.68 ALDH1A1 (0.50) PARP1KDM4EROCK2TNKSROCK1
SCHEMBL4389998 0.66 L3MBTL1 (0.51) CYP2D6KMT2AHSD17B10
SCHEMBL26031894 0.65 PARP1 (0.50) PARP1KDM4ETNKSKMT2AHSD17B10
SCHEMBL14152416 0.65 L3MBTL1 (0.42) MAOBCYP2D6KDM4EAPPKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed