SCHEMBL7142373

SCHEMBL7142373

COc1cccc(C(=O)C(Br)c2ccncc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
CES2 O00748 1/20 0.51
CES1 P23141 1/20 0.51
KMT2A Q03164 1/20 0.50
PARP1 P09874 1/20 0.49
ROCK1 Q13464 5/20 0.47
ROCK2 O75116 4/20 0.47
PRKG1 Q13976 3/20 0.47
CYP2D6 P10635 3/20 0.47
PRKACA P17612 3/20 0.47
GSK3A P49840 3/20 0.47
GSK3B P49841 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CHEK1 O14757 2/20 0.47
RPS6KA5 O75582 2/20 0.47
PRKCG P05129 2/20 0.47
CDK1 P06493 2/20 0.47
RPS6KB1 P23443 2/20 0.47
CDK2 P24941 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6283052 0.99 NPC1 (0.53) NPC1CES2CES1KMT2APARP1
SCHEMBL7144956 0.85 ALDH1A1 (0.55) CES2CES1KMT2ACYP2D6CYP3A4
Bromide SCHEMBL6285575 0.84 ALDH1A1 (0.54) CES2CES1KMT2ACYP2D6CYP3A4
Hydrochloric Acid SCHEMBL11490909 0.83 CES2 (0.51) NPC1CES2CES1KMT2APARP1
SCHEMBL7140563 0.82 CYP1A2 (0.54) NPC1CES2CES1KMT2APARP1
Bromide SCHEMBL5200458 0.82 ROCK2 (0.47) NPC1CES2CES1KMT2APARP1
Bromide SCHEMBL3892616 0.82 ROCK2 (0.47) NPC1CES2CES1KMT2APARP1
Hydrochloric Acid SCHEMBL6708543 0.82 NPC1 (0.53) NPC1CES2CES1KMT2APARP1
Bromide SCHEMBL6284177 0.81 CYP1A2 (0.53) NPC1CES2CES1KMT2APARP1
SCHEMBL7143390 0.81 NT5E (0.52) NPC1KMT2APARP1CHRNA1CHRNG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed