SCHEMBL7143899

SCHEMBL7143899

O=C(O)N1CC[C@@H]2Nc3ccccc3[C@@H]2C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
RBP4 P02753 2/20 0.35
HSPA1A P0DMV8 1/20 0.35
PTPN7 P35236 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ACHE P22303 2/20 0.35
BACE1 P56817 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
BCHE P06276 2/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
TACR3 P29371 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5416718 1.00 LMNA (0.37) LMNATSHRRBP4HSPA1APTPN7
SCHEMBL5416715 1.00 LMNA (0.37) LMNATSHRRBP4HSPA1APTPN7
SCHEMBL5316457 0.89 BCHE (0.39) LMNATSHRRBP4HSPA1APTPN7
SCHEMBL6217421 0.81 MEN1 (0.40) LMNAHSPA1APTPN7TDP1MEN1
SCHEMBL5133257 0.81 GPR119 (0.47)
SCHEMBL28982266 0.79 BACE1 (0.39) LMNATSHRRBP4BACE1ALDH1A1
SCHEMBL21707918 0.79 BACE1 (0.39) LMNATSHRRBP4BACE1ALDH1A1
SCHEMBL3313723 0.79 BACE1 (0.39) LMNATSHRRBP4BACE1ALDH1A1
SCHEMBL14276928 0.76 ALDH1A1 (0.41) ACHEALDH1A1BCHEADRA2AADRA2B
SCHEMBL21871876 0.76 LMNA (0.37) LMNATSHRACHEBCHEPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902684-B1 HEXAHYDRO-PYRIDO(4,3-B)INDOLE DERIVATIVES AS ANTIPSYCHOTIC DRUGS JANSSEN PHARMACEUTICA NV (BE) 2003-04-09 EP disclosed
US-6057325-A HAVE CENTRAL DOPAMINE AND SEROTONIN ANTOGONISTIC ACTIVITY JANSSEN PHARMACEUTIA, N.V. (BE) 2000-05-02 US disclosed