SCHEMBL7144053

SCHEMBL7144053

CCCCC(CC)CNC1CCN([S+]([O-])c2ccc(CNC(=O)c3cccc(OC)c3)s2)CC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
CHRM1 P11229 2/20 0.40
TP53 P04637 1/20 0.37
TSHR P16473 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HPGD P15428 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MCHR1 Q99705 1/20 0.36
EPHX2 P34913 1/20 0.36
PREP P48147 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7145126 0.97 GAA (0.38) GAAMAPTCHRM1TP53TSHR
SCHEMBL7138079 0.86 ALDH1A1 (0.41) GAAMAPTCHRM1TSHRCYP2C9
SCHEMBL7145105 0.85 CHRM1 (0.44) GAAMAPTCHRM1TSHRCYP2C9
SCHEMBL7148318 0.85 CHRM1 (0.43) GAAMAPTCHRM1TSHRCYP2C9
SCHEMBL3480005 0.84 KMT2A (0.51) GAAMAPTCHRM1HPGDPOLB
SCHEMBL7148150 0.84 CHRM1 (0.46) GAACHRM1TSHRCYP2C9CYP2C19
SCHEMBL7138046 0.82 KDM4E (0.38) MAPTTP53TSHRALDH1A1
SCHEMBL7147019 0.82 SMN1; SMN2 (0.39) MAPTTP53TSHRALDH1A1EPHX2
SCHEMBL3479746 0.82 KMT2A (0.48) GAAMAPTCHRM1HPGDPOLB
SCHEMBL3480450 0.82 KMT2A (0.48) GAAMAPTCHRM1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322642-A2 sHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES BEARING BOTH LIPOPHILIC AND IONISABLE MOIETIES AS INHIBITORS OF PROTEIN JUNKINASES Applied Research Systems ARS Holding N.V. (AN) 2003-07-02 EP disclosed
WO-2002026733-A2 sHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES BEARING BOTH LIPOPHILIC AND IONISABLE MOIETIES AS INHIBITORS OF PROTEIN JUNKINASES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2002-04-04 WO disclosed