SCHEMBL7148150

SCHEMBL7148150

COc1cccc(C(=O)NCc2ccc([S+]([O-])N3CCC(NCCO)CC3)s2)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.46
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
PREP P48147 1/20 0.42
HPGD P15428 2/20 0.42
MCHR1 Q99705 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
MMP13 P45452 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7146457 0.89 CHRM1 (0.43) CHRM1CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL7138079 0.89 ALDH1A1 (0.41) CHRM1CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL7145105 0.88 CHRM1 (0.44) CHRM1CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL7148318 0.88 CHRM1 (0.43) CHRM1CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL7146507 0.88 CYP2C9 (0.47) CHRM1CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL7141820 0.88 MCHR1 (0.43) CHRM1ALDH1A1USP2POLBMCHR1
SCHEMBL7143055 0.87 DRD4 (0.47) CHRM1MCHR1MMP13
SCHEMBL7145387 0.87 LMNA (0.45) CHRM1CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL7144671 0.86 MEN1 (0.44) CHRM1CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL7147012 0.86 ALDH1A1 (0.42) CHRM1CYP2C9CYP2C19ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322642-A2 sHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES BEARING BOTH LIPOPHILIC AND IONISABLE MOIETIES AS INHIBITORS OF PROTEIN JUNKINASES Applied Research Systems ARS Holding N.V. (AN) 2003-07-02 EP claimed
WO-2002026733-A2 sHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES BEARING BOTH LIPOPHILIC AND IONISABLE MOIETIES AS INHIBITORS OF PROTEIN JUNKINASES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2002-04-04 WO claimed