SCHEMBL7144469

SCHEMBL7144469

O=C1NC(=O)C2c3ccccc3Oc3cccc1c32

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.40
CYP2C9 P11712 1/20 0.40
ATM Q13315 2/20 0.39
GSK3B P49841 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
POLB P06746 1/20 0.35
USP2 O75604 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9988801 0.81 CYP2C9 (0.37) NISCHCYP2C9ATMGSK3BMAOA
SCHEMBL7142349 0.73 LMNA (0.39) NISCHCYP2C9ATMMAOAMAOB
SCHEMBL29802419 0.72 PARP1 (0.40) NISCHATMMAOAMAOBMEN1
SCHEMBL30312068 0.72 PARP1 (0.40) NISCHATMMAOAMAOBMEN1
SCHEMBL217432 0.72 PARP1 (0.40) NISCHATMMAOAMAOBMEN1
SCHEMBL30785679 0.68 CYP2C9 (0.47) NISCHCYP2C9ATMMAOAMAOB
SCHEMBL7451378 0.68 CYP2C9 (0.38) NISCHCYP2C9ATMMAOAMAOB
SCHEMBL831081 0.67 MAOA (0.37) NISCHCYP2C9ATMMAOAMAOB
SCHEMBL2337529 0.66 GSK3B (0.48) GSK3BMAOAMAOBALDH1A1L3MBTL1
SCHEMBL8516771 0.65 MAOA (0.50) NISCHCYP2C9ATMMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514983-B1 Inhibitors of the nucleic enzyme poly(adenosine 5'-diphospho-ribose)polymerase GUILFORD PHARMACEUTICALS INC. 2003-02-04 US disclosed