SCHEMBL7144589

SCHEMBL7144589

CC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C=O)Cc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSB P07858 3/20 0.61
ALDH1A1 P00352 1/20 0.56
CPA1 P15085 2/20 0.55
CPA2 P48052 2/20 0.55
CPA4 Q9UI42 2/20 0.55
CPB1 P15086 1/20 0.55
ACE2 Q9BYF1 1/20 0.55
MME P08473 2/20 0.53
CMA1 P23946 1/20 0.53
CTRC Q99895 1/20 0.53
CTSL P07711 1/20 0.52
PSMB5 P28074 2/20 0.51
PSMB2 P49721 2/20 0.51
PSMB1 P20618 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13706577 1.00 CTSB (0.61) CTSBALDH1A1CPA1CPA2CPA4
SCHEMBL24178174 0.98 CTSB (0.58) CTSBALDH1A1CPA1CPA2CPA4
SCHEMBL24178168 0.98 CTSB (0.58) CTSBALDH1A1CPA1CPA2CPA4
SCHEMBL24178166 0.92 CTSB (0.56) CTSBALDH1A1CPA1CPA2CPA4
SCHEMBL6248305 0.92 CTSB (0.55) CTSBALDH1A1CPA1CPA2CPA4
SCHEMBL24178171 0.90 CTSB (0.52) CTSBALDH1A1CPA1CPA2CPA4
SCHEMBL24178183 0.90 CTSB (0.52) CTSBALDH1A1CPA1CPA2CPA4
SCHEMBL5572956 0.90 CTSB (0.63) CTSBMMECMA1CTRCCTSL
SCHEMBL20204723 0.90 CTSB (0.63) CTSBMMECMA1CTRCCTSL
SCHEMBL20204725 0.90 CTSB (0.63) CTSBMMECMA1CTRCCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0611756-B1 Alcohol or aldehyde derivatives as cathepsin L inhibitor and bone resorption inhibitor TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-07 EP disclosed
US-5955491-A ADMINISTERING CATHEPSIN L INHIBITOR AND BONE RESORPTION INHIBITOR CONTAINING AN ALCOHOL OR ALDEHYDE DERIVATIVE, OR SALT THEREOF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-09-21 US disclosed
US-5716980-A PROPHYLACTIC, THERAPY FOR OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
US-5639781-A PREVENT REABSORPTION OF BONE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-06-17 US disclosed
US-5498728-A OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-12 US disclosed
EP-0611756-A2 Alcohol or aldehyde derivatives as cathepsin L inhibitor and bone resorption inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-08-24 EP disclosed