SCHEMBL7144739

SCHEMBL7144739

CC(=O)Nc1cc(F)ccc1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
HSD17B10 Q99714 1/20 0.51
GRIK1 P39086 4/20 0.51
CLCN2 P51788 1/20 0.50
HDAC1 Q13547 2/20 0.47
KEAP1 Q14145 1/20 0.46
DYRK1A Q13627 2/20 0.45
PDPK1 O15530 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
MPO P05164 1/20 0.44
GAA P10253 2/20 0.43
KCNK2 O95069 1/20 0.43
STAT1 P42224 1/20 0.43
AVPR2 P30518 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL252578 0.86 KDM4E (0.65) KDM4EHSD17B10HDAC1KEAP1NPC1
SCHEMBL9744446 0.83 GRIK1 (0.49) KDM4EGRIK1CLCN2KEAP1NPC1
SCHEMBL14854686 0.83 SMN1; SMN2 (0.51) KDM4EHSD17B10HDAC1RAB9ACYP2C19
SCHEMBL7848417 0.82 PTPN1 (0.56) GRIK1CLCN2KEAP1NPC1KCNK2
SCHEMBL3810854 0.81 CLCN2 (0.52) KDM4EHSD17B10GRIK1CLCN2KEAP1
SCHEMBL9744178 0.81 KDM4E (0.68) KDM4EGRIK1CLCN2NPC1RAB9A
SCHEMBL12798622 0.81 GRIK1 (0.51) KDM4EGRIK1CLCN2KEAP1NPC1
SCHEMBL13893468 0.80 KDM4E (0.48) KDM4EHDAC1DYRK1APDPK1NPC1
SCHEMBL6891543 0.80 KMT2A (0.55) KDM4EHSD17B10GRIK1CLCN2MEN1
SCHEMBL5490228 0.80 KDM4E (0.57) KDM4EHSD17B10GRIK1HDAC1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4705287-A1 SMALL MOLECULE HUMANIN MIMETICS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-03-11 EP disclosed
WO-2024226731-A1 SMALL MOLECULE HUMANIN MIMETICS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-10-31 WO disclosed
CN-112707845-B Preparation method of dacatinib intermediate 成都伊诺达博医药科技有限公司 2023-04-28 CN disclosed
CN-112707845-A Preparation method of dacomitinib intermediate 成都伊诺达博医药科技有限公司 2021-04-27 CN disclosed
CN-109971210-B Phenolic azo type reactive dye and preparation method thereof 南京林业大学 2021-04-20 CN disclosed
EP-0768301-B1 N-(2-substituted-3-(2-aminoethyl)-1H-indol-5-yl)-amides as new 5-HT1F agonists LILLY CO ELI (US) 2003-04-02 EP disclosed
US-6380201-B1 Methods of treating or ameliorating the symptoms of common cold or allergic rhinitis with serotonin 5-HT1F agonists ELI LILLY AND COMPANY 2002-04-30 US disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
US-6126932-A INSOLUBLE POLYMER BEARING PENDANT SIDE CHAINS, SAID SIDE CHAINS EACH TERMINATING WITH THE 1-(3-(1-PYRROLIDINYL)-PROPYL)-3-ETHYLCARBODIIMIDE MOIETY. ELI LILLY AND COMPANY (US) 2000-10-03 US disclosed
EP-0994109-A2 1-(3-(1-Pyrrolidinyl)propyl)-3-ethylcarbodiimide and a solid phase coupling agent ELI LILLY AND COMPANY (US) 2000-04-19 EP disclosed
EP-0768301-A1 N-(2-substituted-3-(2-aminoethyl)-1H-indol-5-yl)-amides as new 5-HT1F agonists ELI LILLY AND COMPANY (US) 1997-04-16 EP disclosed
US-5302390-A ADMINISTERING TO TREAT THROMBOTIC DISEASES BEECHAM GROUP PLC (GB) 1994-04-12 US disclosed
EP-0297882-B1 HYBRID PLASMINOGEN ACTIVATORS BEECHAM GROUP PLC (GB) 1993-08-25 EP disclosed
WO-1993012795-A1 QUINAZOLIN-4(3H)-ONE DERIVATIVES AS ANTICOCCIDIAL AGENTS GLAZER EDWARD A (US) 1993-07-08 WO disclosed
US-5093364-A 5-FLUOROANTHRANILIC FUNGICIDES SCHERING AGROCHEMICALS LIMITED (GB) 1992-03-03 US disclosed
US-4920224-A CHEMICAL INTERMEDIATES PFIZER INC. (US) 1990-04-24 US disclosed
EP-0360417-A2 Derivatives of 4-fluoroanthranilic acid and their use as fungicides SCHERING AGROCHEMICALS LIMITED (GB) 1990-03-28 EP disclosed
US-4849518-A ANTIPROTOZOA IN POULTRY PFIZER INC. (US) 1989-07-18 US disclosed
EP-0297882-A2 Hybrid plasminogen activators BEECHAM GROUP PLC (GB) 1989-01-04 EP disclosed
US-4762838-A Quinazolin-4(3H)-one derivatives as anticoccidial agents PFIZER INC. (US) 1988-08-09 US disclosed