SCHEMBL7145090

SCHEMBL7145090

CO/N=C(\C)c1cccc(S(N)(=O)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.50
CA2 P00918 12/20 0.48
CA1 P00915 10/20 0.48
CA12 O43570 9/20 0.43
CA9 Q16790 9/20 0.43
CA4 P22748 2/20 0.43
CA14 Q9ULX7 1/20 0.43
F2 P00734 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
STAT3 P40763 1/20 0.42
CA6 P23280 2/20 0.42
CA7 P43166 2/20 0.42
CA13 Q8N1Q1 2/20 0.42
GLO1 Q04760 1/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7145093 1.00 NOS1 (0.50) NOS1CA2CA1CA12CA9
SCHEMBL7142681 0.84 NOS1 (0.47) NOS1CA2CA1CA12CA9
SCHEMBL7142686 0.84 NOS1 (0.47) NOS1CA2CA1CA12CA9
SCHEMBL7143991 0.82 NOS1 (0.54) NOS1CA2CA1CA12CA9
SCHEMBL7143996 0.82 NOS1 (0.54) NOS1CA2CA1CA12CA9
SCHEMBL6814986 0.80 CA2 (0.51) NOS1CA2CA1CA12CA9
SCHEMBL6814989 0.80 CA2 (0.51) NOS1CA2CA1CA12CA9
SCHEMBL7145051 0.79 PPARG (0.54) CA2CA1CA12CA9
SCHEMBL7145050 0.79 PPARG (0.54) CA2CA1CA12CA9
SCHEMBL7613084 0.78 NLRP3 (0.58) CA2CA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964849-B1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY PFIZER (US) 2003-06-04 EP disclosed
EP-1270565-A1 4-Substituted furan-2-sulfonamide and its use in the preparation of sulfonyl urea derivatives PFIZER INC. (US) 2003-01-02 EP disclosed
EP-1270554-A1 Sulfonyl urea derivatives and their use in the control of interleukin-1 activity PFIZER INC. (US) 2003-01-02 EP disclosed
US-6433009-B1 TREATMENT OF AUTOIMMUNE, CARDIOVASCULAR, NERVOUS SYSTEM, GASTROINTESTINAL, RESPIRATORY SYSTEM, AND VIRAL DISORDERS; ANTIDIABETIC, ANTIARTHRITIC, ANTIINFLAMMATORY AND ANTIDEPRESSANT AGENTS PFIZER INC 2002-08-13 US disclosed
US-6166064-A Sulfonyl urea derivatives and their use in the control of interleukin-1 activity PFIZER INC (US) 2000-12-26 US disclosed
EP-0964849-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY PFIZER INC. (US) 1999-12-22 EP disclosed
WO-1998032733-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY PFIZER INC. (US) 1998-07-30 WO disclosed