SCHEMBL7145529

SCHEMBL7145529

[c]1ncccc1-c1ccno1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.38
CYP1A2 P05177 3/20 0.33
CYP19A1 P11511 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2C19 P33261 3/20 0.33
EPHX2 P34913 1/20 0.33
RAB9A P51151 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPC1 O15118 1/20 0.32
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4909130 0.75
SCHEMBL450165 0.72 ALDH1A1 (0.43) RAB9AKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL19439 0.70 NOTUM (0.39) NOTUMCYP1A2CYP19A1RAB9AALDH1A1
SCHEMBL14125002 0.69 NOTUM (0.56) NOTUMCYP1A2CYP19A1CYP2C9CYP2C19
SCHEMBL4590846 0.69 MAPK14 (0.35) CYP19A1RAB9AALDH1A1NPC1
SCHEMBL5797199 0.68 MAPT (0.43) NOTUMCYP1A2CYP2C9CYP2C19RAB9A
SCHEMBL8062583 0.68 NOTUM (0.38) NOTUMCYP1A2CYP19A1CYP2C9CYP2C19
SCHEMBL3397722 0.67 NOTUM (0.35) NOTUMRAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL1393998 0.67
SCHEMBL3766008 0.66 ADRA2A (0.50) CYP1A2CYP19A1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6586441-B2 2-Amino-6-benzylsulfanyl-4-thiophen-2-yl-pyridine-3,5-dicarbo -nitrile as an examplary preferred compound; Alzheimer's and Parkinson's diseases; neuroprotectors; schizophrenia, analgesics; anxiolytic agents; respiratory disorders HOFFMAN-LA ROCHE INC. 2003-07-01 US disclosed