SCHEMBL7147113

SCHEMBL7147113

O=C(c1ccc(OC(F)(F)F)cc1)C(Br)c1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
ABL1 P00519 3/20 0.44
NAMPT P43490 1/20 0.44
TRPV1 Q8NER1 2/20 0.43
TLR7 Q9NYK1 3/20 0.42
TDP1 Q9NUW8 1/20 0.42
GSK3B P49841 1/20 0.41
CCR9 P51686 1/20 0.40
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
EPHX2 P34913 2/20 0.40
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6279968 0.99 ABL1 (0.43) NPC1RAB9AABL1NAMPTTRPV1
SCHEMBL7149547 0.82 GSK3B (0.62) NAMPTTLR7GSK3BEPHX2
SCHEMBL7140563 0.81 CYP1A2 (0.54) NPC1RAB9AGSK3BMEN1KMT2A
Bromide SCHEMBL6284163 0.81 GSK3B (0.60) NAMPTTLR7GSK3BEPHX2
SCHEMBL5527403 0.81 KMT2A (0.46) NPC1RAB9ATRPV1MEN1KMT2A
Bromide SCHEMBL6284177 0.79 CYP1A2 (0.53) NPC1RAB9AGSK3BMEN1KMT2A
SCHEMBL4470958 0.79 LTA4H (0.55) RAB9AGSK3BMEN1KMT2ASMN1; SMN2
Bromide SCHEMBL2795481 0.77 LTA4H (0.53) RAB9AGSK3BMEN1KMT2ASMN1; SMN2
SCHEMBL3537983 0.77 NPC1 (0.59) NPC1RAB9AABL1NAMPTTRPV1
SCHEMBL6695151 0.76 ALDH1A1 (0.36) NAMPTTDP1KMT2ASMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed