SCHEMBL7149547

SCHEMBL7149547

O=C(c1ccc(C(F)(F)F)cc1)C(Br)c1ccncc1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.62
CES2 O00748 2/20 0.54
CES1 P23141 2/20 0.54
PTPN1 P18031 2/20 0.45
KIF11 P52732 1/20 0.43
SRD5A2 P31213 1/20 0.42
PDPK1 O15530 1/20 0.41
TLR7 Q9NYK1 3/20 0.40
SLC6A4 P31645 1/20 0.39
HIF1A Q16665 1/20 0.39
EPAS1 Q99814 1/20 0.39
NAMPT P43490 1/20 0.38
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6284163 0.98 GSK3B (0.60) GSK3BCES2CES1PTPN1KIF11
SCHEMBL7144741 0.86 ALDH1A1 (0.44) GSK3BKIF11SRD5A2HIF1ANAMPT
SCHEMBL3107743 0.85 GSK3B (0.64) GSK3BCES2CES1PTPN1SRD5A2
Bromide SCHEMBL6280874 0.84 ALDH1A1 (0.43) GSK3BKIF11SRD5A2HIF1ANAMPT
SCHEMBL6500852 0.84 CES2 (0.56) GSK3BCES2SRD5A2TLR7
SCHEMBL4470958 0.83 LTA4H (0.55) GSK3BCES2CES1PTPN1
Bromide SCHEMBL6282484 0.83 CES2 (0.55) GSK3BCES2SRD5A2TLR7
SCHEMBL10465540 0.82 GSK3B (0.59) GSK3BCES2CES1PTPN1SRD5A2
Bromide SCHEMBL2795481 0.82 LTA4H (0.53) GSK3BCES2CES1PTPN1
SCHEMBL7147113 0.82 NPC1 (0.44) GSK3BTLR7NAMPTEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed