SCHEMBL7147341

SCHEMBL7147341

O=C(O)OC1=Cc2cc(-c3ccc(Br)cc3)ccc2OC1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RY6 Q15077 5/20 0.44
PTGS2 P35354 15/20 0.43
PTGS1 P23219 8/20 0.43
DRD5 P21918 3/20 0.35
ADRA2A P08913 2/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
DRD1 P21728 1/20 0.35
OPRM1 P35372 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7146217 0.90 PTGS2 (0.44) P2RY6PTGS2PTGS1DRD5ADRA2A
SCHEMBL7148451 0.90 P2RY6 (0.54) P2RY6PTGS2PTGS1DRD5ADRA2A
SCHEMBL7143493 0.89 PTGS2 (0.44) P2RY6PTGS2PTGS1DRD5ADRA2A
SCHEMBL7144214 0.88 PTGS2 (0.54) P2RY6PTGS2PTGS1DRD5DRD3
SCHEMBL7143504 0.83 P2RY6 (0.42) P2RY6PTGS2PTGS1
SCHEMBL6092371 0.81 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6095511 0.81 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL7142450 0.81 PTGS2 (0.40) P2RY6PTGS2PTGS1
SCHEMBL7149865 0.81 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL7142459 0.80 PTGS2 (0.66) P2RY6PTGS2PTGS1DRD5DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977748-B1 SUBSTITUTED BENZOPYRAN DERIVATIVES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2003-03-26 EP claimed