SCHEMBL7147467

SCHEMBL7147467

C=CC(c1ccccc1)(c1ccccc1)c1cccc(C(=O)O)c1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 4/20 0.41
ALOX15 P16050 2/20 0.41
LMNA P02545 1/20 0.39
AKR1C3 P42330 1/20 0.38
NR4A1 P22736 1/20 0.37
NR4A2 P43354 1/20 0.37
NR4A3 Q92570 1/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
MAPT P10636 2/20 0.37
TSHR P16473 1/20 0.37
CDC25B P30305 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
HMGB1 P09429 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10877477 0.80 ALOX15 (0.42) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL29902877 0.78 ALOX15 (0.46) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL28347889 0.78 ALOX15 (0.46) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL9308271 0.78 ALDH1A1 (0.45) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL3650475 0.77 ALDH1A1 (0.43) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL28604177 0.77 ALDH1A1 (0.43) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL8625772 0.74 ALDH1A1 (0.41) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL11540498 0.74 ALDH1A1 (0.41) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL22635 0.72 ALOX15 (0.47) KMT2AALDH1A1ALOX15LMNAAKR1C3
SCHEMBL31229322 0.72 ALOX15 (0.47) KMT2AALDH1A1ALOX15LMNAAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973811-B1 SELF-LIGHT-STABILIZED PHOTOCHROMIC POLYMER, ITS PREPARATION AND ARTICLES CONTAINING SAME CORNING SA (FR) 2003-01-15 EP disclosed
US-6476103-B1 Photochromic organic material, its manufacture and the photochromic articles containing it CORNING INCORPORATED 2002-11-05 US disclosed
US-6316569-B1 RESISTANCE TO PHOTO-FATIGUE; FOR OPHTHALMIC APPLICATIONS CORNING S.A. (FR) 2001-11-13 US disclosed
EP-0973811-A4 SELF-LIGHT-STABILIZED PHOTOCHROMIC POLYMER, ITS PREPARATION AND ARTICLES CONTAINING SAME CORNING SA (FR) 2000-07-12 EP disclosed
EP-0973811-A1 SELF-LIGHT-STABILIZED PHOTOCHROMIC POLYMER, ITS PREPARATION AND ARTICLES CONTAINING SAME CORNING INCORPORATED (US) 2000-01-26 EP disclosed
EP-0931278-A4 PHOTOCHROMIC ORGANIC MATERIAL, ITS MANUFACTURE AND THE PHOTOCHROMIC ARTICLES CONTAINING IT CORNING INC (US) 1999-12-29 EP disclosed
EP-0931278-A1 PHOTOCHROMIC ORGANIC MATERIAL, ITS MANUFACTURE AND THE PHOTOCHROMIC ARTICLES CONTAINING IT CORNING INCORPORATED (US) 1999-07-28 EP disclosed
WO-1998045341-A1 SELF-LIGHT-STABILIZED PHOTOCHROMIC POLYMER, ITS PREPARATION AND ARTICLES CONTAINING SAME CORNING INCORPORATED (US) 1998-10-15 WO disclosed
WO-1998016863-A1 PHOTOCHROMIC ORGANIC MATERIAL, ITS MANUFACTURE AND THE PHOTOCHROMIC ARTICLES CONTAINING IT CORNING INCORPORATED (US) 1998-04-23 WO disclosed