SCHEMBL7147778

SCHEMBL7147778

Cc1ccccc1C(=O)C(Br)c1ccncc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
MAPK1 P28482 1/20 0.47
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ELANE P08246 2/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.40
PLAU P00749 1/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
HSD17B10 Q99714 1/20 0.38
CTNNB1 P35222 1/20 0.38
WNT3A P56704 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6280875 0.98 TYK2 (0.49) TYK2L3MBTL1MAPK1NPC1RAB9A
SCHEMBL7149098 0.83 GAA (0.50) TYK2ELANEKDM4EALDH1A1PLAU
Bromide SCHEMBL6284630 0.82 GAA (0.49) TYK2ELANEKDM4EALDH1A1PLAU
SCHEMBL7148504 0.81 JAK2 (0.50) TYK2MAPK1CYP3A4ELANEALDH1A1
SCHEMBL7149331 0.80 TSHR (0.50) MAPK1NPC1RAB9ACYP1A2CYP2D6
Bromide SCHEMBL6280880 0.79 JAK2 (0.49) TYK2MAPK1CYP3A4ELANEALDH1A1
Bromide SCHEMBL6284643 0.79 TSHR (0.49) MAPK1NPC1RAB9ACYP1A2CYP2D6
SCHEMBL7843732 0.78 KMT2A (0.39) NPC1RAB9AELANEKDM4EALDH1A1
SCHEMBL3115655 0.76 MEN1 (0.52) TYK2L3MBTL1NPC1RAB9ACYP1A2
SCHEMBL27557768 0.75 NPC1 (0.51) TYK2L3MBTL1MAPK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed