SCHEMBL7148308

SCHEMBL7148308

[CH2]C(N)Oc1ccc(-c2nc(C)co2)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.48
ENPP3 O14638 3/20 0.38
ENPP1 P22413 2/20 0.38
PDE4B Q07343 4/20 0.38
PDE4D Q08499 2/20 0.38
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
TGFBR1 P36897 1/20 0.33
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
SCN9A Q15858 1/20 0.33
PPARG P37231 3/20 0.33
PPARA Q07869 3/20 0.33
NOTUM Q6P988 1/20 0.33
STS P08842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28289469 0.77 ENPP3 (0.59) AOC3ENPP3ENPP1PDE4BPDE4D
SCHEMBL6996945 0.76 ENPP3 (0.60) ENPP3ENPP1
SCHEMBL5310580 0.73 ACHE (0.56) AOC3ENPP3ENPP1HDAC1HDAC8
SCHEMBL6328562 0.73 AOC3 (0.61) AOC3ENPP3ENPP1
SCHEMBL8836113 0.73 HDAC1 (0.53) AOC3ENPP3ENPP1PDE4BHDAC1
SCHEMBL2056110 0.72 SCN10A (0.54) AOC3ENPP3ENPP1PDE4BNOTUM
SCHEMBL3085910 0.70 PDE4B (0.51) AOC3ENPP3ENPP1PDE4BHDAC1
SCHEMBL6639205 0.70 HDAC1 (0.51) AOC3ENPP3ENPP1PDE4BHDAC1
SCHEMBL5540418 0.70 PDE4B (0.50) AOC3PDE4BHDAC1HDAC8HDAC6
SCHEMBL2056286 0.70 PDE4B (0.50) AOC3PDE4BHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326861-A1 ALPHA-ARYL ETHANOLAMINES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS Pfizer Products Inc. (US) 2003-07-16 EP disclosed
WO-2002032897-A1 ALPHA-ARYL ETHANOLAMINES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS PFIZER PRODUCTS INC. (US) 2002-04-25 WO disclosed