SCHEMBL7148707

SCHEMBL7148707

CCCCCNC(=O)N1C[C@H](SC(c2ccccc2)(c2ccccc2)c2ccccc2)C[C@H]1COCc1cc(F)c(F)cc1F

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 2/20 0.44
PLA2G4A P47712 2/20 0.36
PLA2G6 O60733 1/20 0.36
ASAH1 Q13510 5/20 0.34
NAMPT P43490 2/20 0.34
LMNA P02545 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPK3 P27361 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SQOR Q9Y6N5 1/20 0.34
CHRM4 P08173 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5407311 0.84 ECE1 (0.51) ECE1PLA2G4APLA2G6CYP2D6
SCHEMBL7146865 0.84 ECE1 (0.51) ECE1PLA2G4APLA2G6CYP2D6
SCHEMBL5400964 0.84 ECE1 (0.44) ECE1PLA2G4APLA2G6CHRM4
SCHEMBL5404278 0.82 ECE1 (0.51) ECE1PLA2G4APLA2G6
SCHEMBL7141469 0.81 ASAH1 (0.39) ECE1ASAH1LMNACYP3A4CYP2D6
SCHEMBL5415467 0.80 ECE1 (0.51) ECE1PLA2G4APLA2G6CYP2D6
SCHEMBL5403789 0.80 ECE1 (0.48) ECE1PLA2G4APLA2G6
SCHEMBL5398705 0.80 PKM (0.39) PLA2G4APLA2G6ASAH1NAMPT
SCHEMBL5407104 0.79 ECE1 (0.47) ECE1PLA2G4APLA2G6CYP2D6
SCHEMBL5407100 0.79 ECE1 (0.47) ECE1PLA2G4APLA2G6CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303486-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
WO-2002008185-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-31 WO disclosed