SCHEMBL7149380

SCHEMBL7149380

Oc1ccc(-c2ccccc2)c2s[c]nc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.41
ALOX5 P09917 2/20 0.40
HPGD P15428 2/20 0.39
ALDH1A1 P00352 1/20 0.39
BCL2L1 Q07817 1/20 0.39
HSD17B10 Q99714 1/20 0.39
COMT P21964 1/20 0.33
ESR2 Q92731 1/20 0.33
HSP90AA1 P07900 1/20 0.33
KDM4E B2RXH2 1/20 0.33
RET P07949 1/20 0.32
FLT1 P17948 1/20 0.32
KDR P35968 1/20 0.32
MAPK14 Q16539 1/20 0.32
RAB9A P51151 3/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
NPC1 O15118 2/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142552 0.76 NQO2 (0.40) HPGDALDH1A1HSD17B10KDM4ERAB9A
SCHEMBL3060568 0.70 PDPK1 (0.47) BACE1ALOX5HPGDALDH1A1BCL2L1
SCHEMBL3060565 0.66 BCAT2 (0.39) BACE1ALOX5ALDH1A1RETFLT1
SCHEMBL4337978 0.66 LIMK1 (0.39) BACE1HPGDALDH1A1BCL2L1HSD17B10
SCHEMBL124933 0.64 PDPK1 (0.44) HPGDALDH1A1HSD17B10COMTKDM4E
SCHEMBL13210303 0.64 BACE1 (0.59) BACE1ALOX5HPGDALDH1A1BCL2L1
SCHEMBL12530867 0.63 COMT (0.73) ALDH1A1COMTHSP90AA1KDM4ERAB9A
SCHEMBL21089511 0.62 HPGD (0.48) HPGDALDH1A1BCL2L1HSD17B10KDM4E
SCHEMBL1889602 0.62 IDO1 (0.65) BACE1ALOX5HPGDALDH1A1BCL2L1
SCHEMBL30669867 0.62 BACE1 (0.56) BACE1ALOX5HPGDALDH1A1BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303272-A2 BENZOTHIAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
WO-2001097786-A2 BENZOTHIAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-12-27 WO disclosed