SCHEMBL7153128

SCHEMBL7153128

C=C(C(=O)OOC(F)(F)F)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.51
ATM Q13315 2/20 0.51
ALDH1A1 P00352 3/20 0.44
TSHR P16473 3/20 0.44
HSD17B10 Q99714 1/20 0.44
CES1 P23141 3/20 0.42
LMNA P02545 2/20 0.41
F2 P00734 1/20 0.41
MAPT P10636 2/20 0.37
ELANE P08246 1/20 0.36
PDK1 Q15118 4/20 0.36
PDK2 Q15119 4/20 0.36
PDK3 Q15120 4/20 0.36
PDK4 Q16654 4/20 0.36
ABCC9 O60706 2/20 0.36
ABCC8 Q09428 2/20 0.36
KCNJ11 Q14654 2/20 0.36
KCNJ8 Q15842 2/20 0.36
ABCB11 O95342 1/20 0.36
CES2 O00748 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9124237 0.82 TDP1 (0.53) TDP1ATMALDH1A1TSHRHSD17B10
SCHEMBL7146887 0.81 TDP1 (0.50) TDP1ATMALDH1A1TSHRHSD17B10
SCHEMBL11074682 0.77 TSHR (0.71) TDP1ALDH1A1TSHRHSD17B10CES1
SCHEMBL28712215 0.75 ATM (0.44) TDP1ATMALDH1A1TSHRCES1
SCHEMBL506074 0.74 TDP1 (0.53) TDP1ATMALDH1A1TSHRHSD17B10
SCHEMBL3875454 0.74 TDP1 (0.58) TDP1ATMALDH1A1TSHRHSD17B10
SCHEMBL906344 0.74 TDP1 (0.46) TDP1ATMALDH1A1CES1LMNA
SCHEMBL30109423 0.73 AKR1C1 (0.54) TDP1ALDH1A1TSHRHSD17B10LMNA
Hydrochloric Acid SCHEMBL31332428 0.73 TDP1 (0.57) TDP1ATMALDH1A1TSHRHSD17B10
SCHEMBL5132603 0.72 TDP1 (0.56) TDP1ATMALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309590-A1 AZAINDOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS ANTITUMOR AGENTS Pharmacia Italia S.p.A. (IT) 2003-05-14 EP disclosed
WO-2001098299-A1 AZAINDOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA ITALIA S.P.A. (IT) 2001-12-27 WO disclosed