Bromide

Bromide

SCHEMBL7154691

Br.CC(=O)O[C@H](CBr)CCNN

nearest known ligand 0.32

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
HRH1 P35367 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TSHR P16473 1/20 0.31
TRPV1 Q8NER1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4922132 0.77 TSHR (0.39) MEN1CYP1A2HRH1KMT2ALMNA
SCHEMBL4922117 0.77 TSHR (0.39) MEN1CYP1A2HRH1KMT2ALMNA
SCHEMBL4930526 0.77 TSHR (0.39) MEN1CYP1A2HRH1KMT2ALMNA
SCHEMBL1116238 0.76
SCHEMBL7753066 0.73 MEN1 (0.36) MEN1CYP1A2HRH1KMT2ALMNA
SCHEMBL764405 0.72 PRKCA (0.42)
SCHEMBL4918612 0.72 ALOX15 (0.41) MEN1CYP1A2HRH1KMT2ALMNA
SCHEMBL4925985 0.72 ALOX15 (0.41) MEN1CYP1A2HRH1KMT2ALMNA
SCHEMBL4918620 0.72 ALOX15 (0.41) MEN1CYP1A2HRH1KMT2ALMNA
SCHEMBL17965847 0.69 PRKCA (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071654-B1 A PROCESS FOR PREPARING CHIRAL (S)-2,3-DISUBSTITUTED-1-PROPYLAMINE DERIVATIVES SAMSUNG FINE CHEMICALS CO LTD (KR) 2003-10-22 EP disclosed
US-6417403-B1 AMINATION OF 3,4-DISUBSTITUTED-1-BUTANECARBONYL DERIVATIVE THROUGH CURTIUS OR HOFMAN REARRANGEMENT; SALT FORMATION, CARBAMYLATION SAMSUNG FINE CHEMICALS CO., LTD. (KR) 2002-07-09 US disclosed
EP-1071654-A1 A PROCESS FOR PREPARING CHIRAL (S)-2,3-DISUBSTITUTED-1-PROPYLAMINE DERIVATIVES Samsung Fine Chemicals Co., Ltd. (KR) 2001-01-31 EP disclosed
WO-1999052855-A1 A PROCESS FOR PREPARING CHIRAL (S)-2,3-DISUBSTITUTED-1-PROPYLAMINE DERIVATIVES SAMSUNG FINE CHEMICALS CO., LTD. (KR) 1999-10-21 WO disclosed