SCHEMBL715873

SCHEMBL715873

CC(NC(=O)O)c1cc2cccc(Br)c2nc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
LMNA P02545 1/20 0.38
KDR P35968 2/20 0.36
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
PDE2A O00408 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
GPR139 Q6DWJ6 2/20 0.34
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL844461 0.87 MAPT (0.46) HTTKDRMEN1NPC1GAA
SCHEMBL5302 0.87 GPR139 (0.39) MEN1NPC1GAAMAPTRAB9A
SCHEMBL716685 0.77 L3MBTL1 (0.34) MEN1KMT2AL3MBTL1PDE2AGPR139
SCHEMBL721702 0.74 KDR (0.41) HTTKDRMEN1NPC1GAA
SCHEMBL721701 0.74 KDR (0.41) HTTKDRMEN1NPC1GAA
SCHEMBL716039 0.74 ALDH1A1 (0.31) ALDH1A1
SCHEMBL716038 0.74 ALDH1A1 (0.31) ALDH1A1
SCHEMBL864754 0.73 PIK3CD (0.38) L3MBTL1PDE2AGPR139
SCHEMBL717883 0.73 SOS1 (0.36) ALDH1A1MAPTPDE2A
SCHEMBL713467 0.72 TSHR (0.43) HTTLMNAKDRMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403847-B1 TRIAZINE DERIVATIVES AS KINASE INHIBITORS UCB BIOPHARMA SPRL (BE) 2016-03-02 EP disclosed
US-8785628-B2 Triazine derivatives as kinase inhibitors UCB PHARMA, S.A. (BE) 2014-07-22 US disclosed
US-20120053167-A1 Triazine Derivatives as Kinase Inhibitors UCB PHARMA, S.A. (BE) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053167-A1 Triazine Derivatives as Kinase Inhibitors MAP3K15, PI4KA, MAP3K20 HTT 1681/4885LMNA 4722/4885KDR 437/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.