SCHEMBL7160899

SCHEMBL7160899

CC(C)(C)OC(=O)N[C@@H](Cc1ccc2c(c1)NC(=O)[C@@H](CCC(=O)Nc1nc3ccccc3[nH]1)O2)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.49
ACE P12821 2/20 0.42
ITGB3 P05106 5/20 0.41
ITGAV P06756 5/20 0.41
IDO1 P14902 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
BCHE P06276 1/20 0.39
CCKAR P32238 1/20 0.39
CCKBR P32239 1/20 0.39
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PIN1 Q13526 2/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3050522 0.93 PTPN1 (0.51) PTPN1ACEITGB3ITGAVIDO1
SCHEMBL7478478 0.93 PTPN1 (0.41) PTPN1ITGB3ITGAVNPC1RAB9A
SCHEMBL7165492 0.87 PTPN1 (0.44) PTPN1ITGB3ITGAVNPC1RAB9A
SCHEMBL7163716 0.86 ACE (0.41) PTPN1ACEITGB3ITGAVIDO1
SCHEMBL7163504 0.86 ACE (0.41) PTPN1ACEITGB3ITGAVIDO1
SCHEMBL7478067 0.86 PTPN1 (0.44) PTPN1ITGB3ITGAVNPC1RAB9A
SCHEMBL7161074 0.84 NPC1 (0.43) NPC1RAB9AHTTSMN1; SMN2
SCHEMBL8324174 0.84 ITGB3 (0.44) ITGB3ITGAVNPC1RAB9AHTT
SCHEMBL7164117 0.84 PTPN1 (0.55) PTPN1ACEITGB3ITGAVIDO1
SCHEMBL7168844 0.83 ITGAV (0.45) ITGB3ITGAVNPC1RAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6559144-B2 Integrin inhibitors used to treat circulatory disorders, for thrombosis, myocardial infarct, coronary heart disease, arteriosclerosis, osteoporosis, pathological processes maintained or propagated by angiogenesis and tumor therapy MERCK PATENT GESELLSCHAFT MIT (DE) 2003-05-06 US disclosed
EP-0964856-B1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 2002-10-09 EP disclosed
US-20010021709-A1 Bicyclic amino acids MERCK PATENT GESELLSCHAFT MIT BESCHRANKT PATENTS (DE) 2001-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010021709-A1 Bicyclic amino acids ITGA1, ITGB1, ITGB2 PTPN1 2528/4885ACE 3019/4885ITGB3 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.