SCHEMBL7162986

SCHEMBL7162986

O=C(Nc1ccc(NC(=S)NCCSc2cccc(Br)c2)cc1)c1ccco1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
KMT2A Q03164 8/20 0.52
MEN1 O00255 6/20 0.52
MAPT P10636 4/20 0.52
HTT P42858 2/20 0.52
GAA P10253 2/20 0.52
BLM P54132 1/20 0.52
POLB P06746 3/20 0.50
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
HPGD P15428 4/20 0.48
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 2/20 0.47
RECQL P46063 1/20 0.47
USP2 O75604 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7865724 0.87 RAB9A (0.70) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6817086 0.80 KDM4E (0.51) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6816108 0.80 KMT2A (0.48) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6817088 0.80 MAPT (0.49) RAB9ASMN1; SMN2KMT2AMEN1MAPT
SCHEMBL6816313 0.78 MAPT (0.46) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL7158954 0.78 RAB9A (0.67) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL7163839 0.76 NPC1 (0.62) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL7167224 0.75 RAB9A (0.74) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL7159264 0.73 KMT2A (0.67) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL7157761 0.72 RAB9A (0.60) NPC1RAB9ASMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6555561-B2 N-(5-((((5-Chloro-2,4-dimethoxyphenyl)amino)thioxomethyl)-amino)-2 -pyridinyl)-2-methylbenzamide, for example; inhibiting replication of a herpes virus WYETH 2003-04-29 US disclosed