SCHEMBL7166169

SCHEMBL7166169

COC(=O)N1C[C@@H]2CCC(CNCc3cccc(C)c3)CC2CC1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 6/20 0.43
NPC1 O15118 1/20 0.36
GRIN2B Q13224 2/20 0.36
GRM5 P41594 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CCR5 P51681 1/20 0.35
BCHE P06276 1/20 0.35
CFD P00746 1/20 0.35
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7171997 0.90 CXCR4 (0.40) CXCR4ALDH1A1
SCHEMBL7168130 0.88 KMT2A (0.38) CXCR4NPC1ALDH1A1
SCHEMBL7165958 0.84 AGTR2 (0.41)
SCHEMBL7170826 0.83 CXCR4 (0.40) CXCR4GRIN2B
SCHEMBL7162414 0.80 DPP4 (0.41) ALDH1A1CFD
SCHEMBL7141654 0.80 LTC4S (0.37) GRM5ALDH1A1BRD4
SCHEMBL7168153 0.80 GRIN2B (0.46) CXCR4GRIN2BALDH1A1BCHEBRD4
SCHEMBL6484834 0.75 TACR1 (0.41) GRIN2BALDH1A1BCHE
SCHEMBL6326567 0.74 NR1H2 (0.40) ALDH1A1
SCHEMBL7162429 0.73 TSHR (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082856-A1 ISOQUINOLINE-3-CARBOXYLIC ACID DERIVATIVES AS EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2003-10-09 WO disclosed