SCHEMBL7167167

SCHEMBL7167167

Cc1c(-c2ccc(O)cc2)ccc(C#N)c1I

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 6/20 0.50
AR P10275 4/20 0.41
MMP3 P08254 1/20 0.40
CYP19A1 P11511 2/20 0.37
ESR1 P03372 5/20 0.37
USP7 Q93009 3/20 0.37
SENP1 Q9P0U3 1/20 0.36
CA12 O43570 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CA6 P23280 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
ESRRB O95718 1/20 0.35
ESRRA P11474 1/20 0.35
PGR P06401 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450852 0.76 ESR2 (0.68) ESR2ARMMP3ESR1SENP1
SCHEMBL4421994 0.73 MMP3 (0.44) ARMMP3CA12CA2CA3
SCHEMBL12801483 0.71 SENP1 (0.43) ESR2ESR1USP7SENP1
SCHEMBL13807442 0.70 TSHR (0.43) AR
SCHEMBL14173712 0.69 AR (0.50) ESR2ARMMP3ESR1USP7
SCHEMBL2785589 0.68 AR (0.57) ESR2ARMMP3ESR1
SCHEMBL1532429 0.67 ESR2 (1.00) ESR2ARMMP3CYP19A1ESR1
SCHEMBL14675564 0.67 ESR2 (0.43) ESR2ARMMP3CYP19A1ESR1
SCHEMBL4667162 0.67 ESR2 (0.59) ESR2ARMMP3CYP19A1ESR1
SCHEMBL4650125 0.66 ESR1 (0.48) ESR2ARESR1USP7SENP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370546-A2 NOVEL AMINES AS HISTAMINE-3 RECEPTOR LIGANDS AND THEIR THERAPEUTIC APPLICATIONS Abbott Laboratories (US) 2003-12-17 EP disclosed
WO-2002074758-A2 NOVEL AMINES AS HISTAMINE-3 RECEPTOR LIGANDS AND THEIR THERAPEUTIC APPLICATIONS ABBOTT LABORATORIES (US) 2002-09-26 WO disclosed