SCHEMBL7168100

SCHEMBL7168100

O=[C]c1cc(Br)c(OCCc2ccccc2)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
THRA P10827 4/20 0.44
THRB P10828 4/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
FFAR1 O14842 1/20 0.42
RHEB Q15382 1/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
ESR1 P03372 1/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38
AR P10275 1/20 0.38
LTA4H P09960 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7161992 0.92 THRA (0.43) THRATHRBFFAR1RHEBMAOA
SCHEMBL7164250 0.91 FFAR1 (0.44) THRATHRBFFAR1
SCHEMBL7163248 0.90 FFAR1 (0.43) THRATHRBFFAR1
SCHEMBL9218172 0.90 FFAR1 (0.43) THRATHRBFFAR1
SCHEMBL7165516 0.84 THRA (0.57) THRATHRBCA12CA1CA2
SCHEMBL7168103 0.78 ALDH1A1 (0.50) THRATHRBCA12CA1CA2
SCHEMBL12370681 0.75 ALDH1A1 (0.48) THRATHRBCA12CA1CA2
SCHEMBL8995355 0.75 NPC1 (0.62) CA12CA1CA2CA7CA9
SCHEMBL526539 0.73 LTA4H (0.45) THRATHRBCA12CA1CA2
SCHEMBL9099031 0.73 FFAR1 (0.53) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1044002-A4 METHODS FOR TREATMENT OF DISORDERS OF CARDIAC CONTRACTILITY UNIV JOHNS HOPKINS (US) 2003-05-02 EP disclosed
EP-1044002-A1 METHODS FOR TREATMENT OF DISORDERS OF CARDIAC CONTRACTILITY JOHNS HOPKINS UNIVERSITY (US) 2000-10-18 EP disclosed
WO-1999024038-A1 METHODS FOR TREATMENT OF DISORDERS OF CARDIAC CONTRACTILITY JOHNS HOPKINS UNIVERSITY (US) 1999-05-20 WO disclosed