Tonabersat

Tonabersat

SCHEMBL7169677

CC(=O)c1ccc2c(c1)[C@H](NC(=O)c1ccc(F)c(Cl)c1)[C@@H](O)C(C)(C)O2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 5/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tonabersat SCHEMBL29377931 1.00 ABCC9 (0.62) ABCC9
Tonabersat SCHEMBL260661 1.00 ABCC9 (0.62) ABCC9
Tonabersat SCHEMBL29373962 1.00 ABCC9 (0.62) ABCC9
Tonabersat SCHEMBL5917016 1.00 ABCC9 (0.62) ABCC9
Tonabersat SCHEMBL29717099 1.00 ABCC9 (0.62) ABCC9
Tonabersat SCHEMBL29370960 0.93 ABCC9 (0.54) ABCC9
Tonabersat SCHEMBL15973365 0.93 ABCC9 (0.54) ABCC9
SCHEMBL7044135 0.89 ABCC9 (0.59) ABCC9
SCHEMBL15546692 0.88 ABCC9 (0.48) ABCC9
SCHEMBL15546693 0.88 ABCC9 (0.48) ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908860-A Bicyclic compounds with pharmaceutical activity SMITHKLINE BEECHAM PLC, (GB) 1999-06-01 US claimed
EP-0673373-A1 BICYCLIC COMPOUNDS WITH PHARMACEUTICAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-09-27 EP claimed
WO-1994013656-A1 BICYCLIC COMPOUNDS WITH PHARMACEUTICAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1994-06-23 WO claimed
US-20160318892-A1 PRODRUG COMPOUNDS PROXIMAGEN LIMITED (GB) 2016-11-03 US disclosed
US-20160318892-A1 PRODRUG COMPOUNDS PROXIMAGEN LIMITED (GB) 2016-11-03 US disclosed
US-20160318892-A1 PRODRUG COMPOUNDS PROXIMAGEN LIMITED (GB) 2016-11-03 US disclosed
WO-2015097461-A1 PRODRUG COMPOUNDS PROXIMAGEN LIMITED (GB) 2015-07-02 WO disclosed
EP-1114821-B1 Benzopyrans and their use as therapeutic agents SMITHKLINE BEECHAM PLC (GB) 2003-09-17 EP disclosed
WO-2002042285-A1 NOVEL PROCESS FOR THE PREPARATION OF 4-BENZOYLAMINO CHROMAN DERIVATIVES SMITHKLINE BEECHAM P.L.C. (GB) 2002-05-30 WO disclosed
EP-0764157-B1 BENZOPYRANS AND THEIR USE AS THERAPEUTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 2002-01-02 EP disclosed
EP-1114821-A1 Benzopyrans and their use as therapeutic agents SMITHKLINE BEECHAM PLC (GB) 2001-07-11 EP disclosed
US-5908860-A Bicyclic compounds with pharmaceutical activity SMITHKLINE BEECHAM PLC, (GB) 1999-06-01 US disclosed
EP-0764157-A1 BENZOPYRANS AND THEIR USE AS THERAPEUTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-03-26 EP disclosed
WO-1995034545-A1 BENZOPYRANS AND THEIR USE AS THERAPEUTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 1995-12-21 WO disclosed
EP-0673373-A1 BICYCLIC COMPOUNDS WITH PHARMACEUTICAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-09-27 EP disclosed
WO-1994013656-A1 BICYCLIC COMPOUNDS WITH PHARMACEUTICAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1994-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160318892-A1 PRODRUG COMPOUNDS SCN1B, CACNA1E, SCN2B ABCC9 370/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.